IS6922A
Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
Abstract
The present invention provides compounds and pharmaceutical compositions that act as antagonists at metabotropic glutamate receptors, and that are useful for treating neurological diseases and disorders. Method of preparing the compounds also are disclosed.
Term
No projected expiry on record.
- Priority
- Filed and published
- Today
95 members in 31 offices
Priority claims7
| Document | Office | Kind | Date |
|---|---|---|---|
| 26984701 | United States of America | P | |
| 26984701 | United States of America | P | |
| 0204689 | United States of America | W | |
| 0204689 | United States of America | W | |
| PCTUS0204689 | – | – | – |
| US20010269847P | – | – | – |
| WO2002US04689 | – | – | – |
Members95
| Document | Office | Kind | |
|---|---|---|---|
| CA2381975A1 | Canada | A1 | |
| WO0112627A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU6782400A | Australia | A | |
| IS6275A | Iceland | A | |
| NO20020823D0 | Norway | D0 | |
| NO20020823L | Norway | L | |
| KR20020038731A | Republic of Korea | A | |
| EP1210344A1 | European Patent Office (EPO) | A1 | |
| CZ2002599A3 | Czechia | A3 | |
| SK2512002A3 | Slovakia | A3 | |
| BR0013427A | Brazil | A | |
| CA2438991A1 | Canada | A1 | |
| WO02068417A2 | World Intellectual Property Organization (WIPO) | A2 | |
| IL148157A0 | Israel | A0 | |
| IL148157D0 | Israel | D0 | |
| CN1379775A | China | A | |
| WO02068417A3 | World Intellectual Property Organization (WIPO) | A3 | |
| HU0202757A2 | Hungary | A2 | |
| HUP0202757A2 | Hungary | A2 | |
| BG106493A | Bulgaria | A | |
| JP2003507378A | Japan | A | |
| HK1047929A | Hong Kong, China | A | |
| HK1047929A1 | Hong Kong, China | A1 | |
| US2003055085A1 | United States of America | A1 | |
| EE200200079A | Estonia | A | |
| ZA200201358B | South Africa | B | |
| IS6922AThis record | Iceland | A | |
| NO20033711D0 | Norway | D0 | |
| NO20033711L | Norway | L | |
| KR20030088434A | Republic of Korea | A | |
| PL353825A1 | Poland | A1 | |
| US6660753B2 | United States of America | B2 | |
| EP1379525A2 | European Patent Office (EPO) | A2 | |
| NZ517221A | New Zealand | A | |
| MXPA02001764A | Mexico | A | |
| IL157491A0 | Israel | A0 | |
| IL157491D0 | Israel | D0 | |
| MXPA03007513A | Mexico | A | |
| HK1060559A1 | Hong Kong, China | A1 | |
| BR0207390A | Brazil | A | |
| ZA200306493B | South Africa | B | |
| JP2004536037A | Japan | A | |
| AU780191B2 | Australia | B2 | |
| RU2003128535A | Russian Federation | A | |
| PL369598A1 | Poland | A1 | |
| US2005154027A1 | United States of America | A1 | |
| CN1649865A | China | A | |
| EP1582519A2 | European Patent Office (EPO) | A2 | |
| EP1210344B1 | European Patent Office (EPO) | B1 | |
| AT307129T | Austria | T | |
| ATE307129T1 | Austria | T1 | |
| UA74419C2 | Ukraine | C2 | |
| EP1582519A3 | European Patent Office (EPO) | A3 | |
| DE60023318D1 | Germany | D1 | |
| DK1210344T3 | Denmark | T3 | |
| HU0202757A3 | Hungary | A3 | |
| HUP0202757A3 | Hungary | A3 | |
| ES2250177T3 | Spain | T3 | |
| JP2006143746A | Japan | A | |
| UA75871C2 | Ukraine | C2 | |
| JP3790472B2 | Japan | B2 | |
| EP1679313A2 | European Patent Office (EPO) | A2 | |
| JP2006182789A | Japan | A | |
| DE60023318T2 | Germany | T2 | |
| EP1679313A3 | European Patent Office (EPO) | A3 | |
| US2006189661A1 | United States of America | A1 | |
| US7112595B2 | United States of America | B2 | |
| NO322460B1 | Norway | B1 | |
| CN1853630A | China | A | |
| NZ527691A | New Zealand | A | |
| RU2296127C2 | Russian Federation | C2 | |
| CN1313465C | China | C | |
| IL148157A | Israel | A | |
| CN1332959C | China | C | |
| RU2296127C9 | Russian Federation | C9 | |
| AU2002306517B2 | Australia | B2 | |
| EP1379525B1 | European Patent Office (EPO) | B1 | |
| AT375340T | Austria | T | |
| ATE375340T1 | Austria | T1 | |
| DE60222872D1 | Germany | D1 | |
| PT1379525E | Portugal | E | |
| DK1379525T3 | Denmark | T3 | |
| SI1379525T1 | Slovenia | T1 | |
| ES2292830T3 | Spain | T3 | |
| RU2319701C2 | Russian Federation | C2 | |
| KR100838447B1 | Republic of Korea | B1 | |
| DE60222872T2 | Germany | T2 | |
| NO326105B1 | Norway | B1 | |
| KR100875222B1 | Republic of Korea | B1 | |
| BG65586B1 | Bulgaria | B1 | |
| IS2564B | Iceland | B | |
| CY1105253T1 | Cyprus | T1 | |
| JP4519404B2 | Japan | B2 | |
| CA2438991C | Canada | C | |
| CY1107005T1 | Cyprus | T1 |
Numbers
- Publication, DOCDB
- 6922
- Publication, EPODOC
- IS6922
- Application
- 6922
- Application, DOCDB
- 6922
- Application, EPODOC
- IS20030006922
Titles2
- Icelandic
- Heterófjölhringjaefnasambönd og notkun þeirra semmetabótrópísk mótlyf gegn glútamat viðtökum
- English
- Hetero-polycyclic compounds and their use as a metabotropic anti-glutamate receptor antagonist
Classification
- CPC, 28
- C07D213/75
- C07D413/14
- A61P3/08
- C07D213/55
- A61P9/10
- C07D213/78
- A61P17/02
- C07D213/79
- A61P25/00
- C07D231/12
- A61P25/02
- C07D233/56
- A61P25/04
- C07D249/08
- A61P25/06
- C07D401/04
- A61P25/08
- C07D405/04
- A61P25/14
- C07D405/14
- A61P25/16
- C07D413/04
- A61P25/18
- A61P25/22
- C07D417/04
- A61P25/28
- A61P29/00
- A61P43/00
- IPC, 24
- A61K31 443
- C07D413 00
- A61K31 4439
- A61K31 444
- A61P25 00
- A61P25 04
- A61P25 06
- A61P25 08
- A61P25 14
- A61P25 16
- A61P25 18
- A61P25 22
- A61P25 28
- C07D213 55
- C07D213 75
- C07D213 78
- C07D213 79
- C07D401 04
- C07D405 04
- C07D405 14
- C07D413 04
- C07D413 14
- C07D417 04
- C07D521 00