IS5722A
PYRROLO 2,3-d]PYRIMIDINE COMPOUNDS
Abstract
A compound of formula (I) wherein R<1>, R<2> and R<3> are as defined in the formula which are inhibitors of the enzyme protein tyrosine kinases such as Janus Kinase 3 and as such are useful therapy as immunosuppresive agents for organ transplants, lupus, multiple sclesoris, rheumatoid arthritis, psoriasis, Type I diabetes and complications from diabetes, cancer, asthma, atopic dermatitis, autoimmune thyroid disorders, ulcerative colitis, Crohn's disease, Alzheimer's disease, Leukemia and other autoimmune diseases.
Term
Term ended
Projected expiry passed 21 November 2020, 5.8 years ago.
- Priority
- Filed and published
- Projected expiry
- Today
150 members in 49 offices
Priority claims7
| Document | Office | Kind | Date |
|---|---|---|---|
| 8988698 | United States of America | P | |
| 8988698 | United States of America | P | |
| 9901110 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| 9901110 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| PCTIB9901110 | – | – | – |
| US19980089886P | – | – | – |
| WO1999IB01110 | – | – | – |
Members150
| Document | Office | Kind | |
|---|---|---|---|
| CA2335186A1 | Canada | A1 | |
| CA2335492A1 | Canada | A1 | |
| WO9965908A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO9965909A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU3951899A | Australia | A | |
| AU4054599A | Australia | A | |
| PE20000639A1 | Peru | A1 | |
| PE20000698A1 | Peru | A1 | |
| PA8474101A1 | Panama | A1 | |
| IS5721A | Iceland | A | |
| IS5722AThis record | Iceland | A | |
| GT199900090A | Guatemala | A | |
| GT199900091A | Guatemala | A | |
| NO20006453D0 | Norway | D0 | |
| NO20006454D0 | Norway | D0 | |
| ZA994003B | South Africa | B | |
| ZA994004B | South Africa | B | |
| ID26698A | Indonesia | A | |
| NO20006453L | Norway | L | |
| NO20006454L | Norway | L | |
| NO20050201L | Norway | L | |
| BR9911365A | Brazil | A | |
| TR200003719T2 | Türkiye | T2 | |
| TR200003720T2 | Türkiye | T2 | |
| EP1087970A1 | European Patent Office (EPO) | A1 | |
| EP1087971A1 | European Patent Office (EPO) | A1 | |
| BR9912171A | Brazil | A | |
| ID27595A | Indonesia | A | |
| HN1999000083A | Honduras | A | |
| EA200001188A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200001203A1 | Eurasian Patent Organization (EAPO) | A1 | |
| KR20010053004A | Republic of Korea | A | |
| KR20010053005A | Republic of Korea | A | |
| AR016498A1 | Argentina | A1 | |
| AR016499A1 | Argentina | A1 | |
| CN1305479A | China | A | |
| CN1305480A | China | A | |
| NO20050202L | Norway | L | |
| BG105122A | Bulgaria | A | |
| HRP20000885A2 | Croatia | A2 | |
| HRP20000886A2 | Croatia | A2 | |
| AP1021A | African Regional Intellectual Property Organization (ARIPO) | A | |
| HU0102574A2 | Hungary | A2 | |
| HUP0102574A2 | Hungary | A2 | |
| BG105129A | Bulgaria | A | |
| PL345118A1 | Poland | A1 | |
| PL345123A1 | Poland | A1 | |
| HK1036800A1 | Hong Kong, China | A1 | |
| HK1036801A1 | Hong Kong, China | A1 | |
| HU0102574A3 | Hungary | A3 | |
| HUP0102574A3 | Hungary | A3 | |
| IL139586D0 | Israel | D0 | |
| IL139598D0 | Israel | D0 | |
| US2002019526A1 | United States of America | A1 | |
| HU0103472A2 | Hungary | A2 | |
| HUP0103472A2 | Hungary | A2 | |
| CZ20004726A3 | Czechia | A3 | |
| CZ20004727A3 | Czechia | A3 | |
| JP2002518393A | Japan | A | |
| JP2002518394A | Japan | A | |
| SK18982000A3 | Slovakia | A3 | |
| SK18992000A3 | Slovakia | A3 | |
| TW505646B | Taiwan Province of China | B | |
| HU0103472A3 | Hungary | A3 | |
| HUP0103472A3 | Hungary | A3 | |
| AU758427B2 | Australia | B2 | |
| YU78500A | Yugoslavia, later Serbia and Montenegro (until 2006) | A | |
| YU79700A | Yugoslavia, later Serbia and Montenegro (until 2006) | A | |
| AP1157A | African Regional Intellectual Property Organization (ARIPO) | A | |
| TW542834B | Taiwan Province of China | B | |
| US6610847B2 | United States of America | B2 | |
| PA8476001A1 | Panama | A1 | |
| AU2003234874A1 | Australia | A1 | |
| CO5320601A1 | Colombia | A1 | |
| US6635762B1 | United States of America | B1 | |
| CN1125070C | China | C | |
| US2003212273A1 | United States of America | A1 | |
| CN1128800C | China | C | |
| NZ508034A | New Zealand | A | |
| UA63013C2 | Ukraine | C2 | |
| KR100415791B1 | Republic of Korea | B1 | |
| JP3497823B2 | Japan | B2 | |
| UA64792C2 | Ukraine | C2 | |
| US2004058922A1 | United States of America | A1 | |
| EP1087970B1 | European Patent Office (EPO) | B1 | |
| NZ518444A | New Zealand | A | |
| AT265458T | Austria | T | |
| ATE265458T1 | Austria | T1 | |
| DE69916833D1 | Germany | D1 | |
| PT1087970E | Portugal | E | |
| OA11571A | African Intellectual Property Organization (OAPI) | A | |
| OA11572A | African Intellectual Property Organization (OAPI) | A | |
| EP1087971B1 | European Patent Office (EPO) | B1 | |
| AT270673T | Austria | T | |
| ATE270673T1 | Austria | T1 | |
| DK1087970T3 | Denmark | T3 | |
| DE69918552D1 | Germany | D1 | |
| AU2003234874B2 | Australia | B2 | |
| KR100452054B1 | Republic of Korea | B1 | |
| DK1087971T3 | Denmark | T3 |
Showing 100 of 150
Numbers
- Publication, DOCDB
- 5722
- Publication, EPODOC
- IS5722
- Application
- 5722
- Application, DOCDB
- 5722
- Application, EPODOC
- IS20000005722
Titles2
- Icelandic
- Pýróló [2,3-dl]pírimídín efnasambönd
- English
- Pyrolo [2,3-dl] pyrimidine compounds
Classification
- CPC, 16
- C07D487/04
- A61P1/04
- A61P11/06
- A61P17/04
- A61P19/02
- A61P25/00
- A61P25/18
- A61P25/28
- A61P29/00
- A61P35/00
- A61P35/02
- A61P37/00
- A61P37/06
- A61P5/14
- A61P5/16
- A61P3/10
- IPC, 18
- A61K31 505
- A61K31 519
- A61K31 5377
- A61K31 55
- A61P1 04
- A61P3 10
- A61P5 14
- A61P11 06
- A61P17 04
- A61P19 02
- A61P25 00
- A61P25 28
- A61P29 00
- A61P35 00
- A61P35 02
- A61P37 06
- C07D487 04
- C07D519 00