Stabilized benzimidazole derivative and composition
Abstract
A stabilized physiologically active benzimidazole derivative having the formula (I): wherein R¹ is hydrogen atom, an alkyl group having 1 to 8 carbon atoms, a fluoroalkyl group having 1 to 6 carbon atoms, a cycloalkyl group, phenyl group or an aralkyl group, R² is hydrogen atom or a lower alkyl group, or R¹ and R² together with the adjacent nitrogen atom form a ring, and each of R3a, R3b, R4a, R4b and R4c independently is hydrogen atom, a halogen atom, a flouroalkyl group having 1 to 6 carbon atoms, a lower alkyl group, a lower alkoxy group, a lower alkoxycarbonyl group or an amino group. The stabilized benzimdazole derivative is in amorphous form or present in contact with a basic material.

Term
Term ended
Projected expiry passed 2 June 2007, 19.3 years ago.
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1 sheet
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Every citation, both ways
| Document | Relation | Office | Category | Cited during |
|---|---|---|---|---|
| EP0204215A1 | Cites | European Patent Office (EPO) | XP | Search report |
| EP0218336A2 | Cites | European Patent Office (EPO) | XP | Search report |
19 members in 8 offices
Priority claims15
| Document | Office | Kind | Date |
|---|---|---|---|
| 12898886 | Japan | A | |
| 12898886 | Japan | A | |
| 12898886 | Japan | – | |
| 12898986 | Japan | A | |
| 12898986 | Japan | A | |
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| 16061286 | Japan | A | |
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| 16061286 | – | – | – |
| JP19860128988 | – | – | – |
| JP19860128989 | – | – | – |
| JP19860160612 | – | – | – |
Members19
| Document | Office | Kind | |
|---|---|---|---|
| AU7369987A | Australia | A | |
| EP0248634A2 | European Patent Office (EPO) | A2 | |
| JPS62283964A | Japan | A | |
| JPS62283965A | Japan | A | |
| JPS6314773A | Japan | A | |
| EP0248634A3This record | European Patent Office (EPO) | A3 | |
| KR880000405A | Republic of Korea | A | |
| AU619444B2 | Australia | B2 | |
| AU1858192A | Australia | A | |
| EP0248634B1 | European Patent Office (EPO) | B1 | |
| DE3786606D1 | Germany | D1 | |
| US5294439A | United States of America | A | |
| DE3786606T2 | Germany | T2 | |
| AR246515A1 | Argentina | A1 | |
| ES2058114T3 | Spain | T3 | |
| JPH0791273B2 | Japan | B2 | |
| JPH0791274B2 | Japan | B2 | |
| JPH0791275B2 | Japan | B2 | |
| KR950011414B1 | Republic of Korea | B1 |
42 legal events, as 4 offices reported them to INPADOC
Over the term
Point at a mark for the eventEvents
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|---|---|---|---|
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Announcement of lapse in spainLapsedFD2A | FD2A | ES | |
| Notification of lapseLapsedST | ST | FR | |
| Se: european patent has lapsedLapsedEUG | EUG | EP | |
| Nl: lapsed or anulled due to non-payment of the annual feeLapsedNLV4 | NLV4 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Patent ceasedCeasedPL | PL | CH | |
| Gb: european patent ceased through non-payment of renewal feeCeasedGBPC | GBPC | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Be: lapsedLapsedBERE | BERE | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Se: european patent in force in swedenEAL | EAL | EP | |
| Definitive protectionFG2A | FG2A | ES | |
| No opposition filedOpposition26N | 26N | EP | |
| No opposition filed within time limitOppositionORIGINAL CODE: 0009261PLBE | PLBE | EP | |
| Information on the status of an ep patent application or granted ep patentGrantedSTATUS: NO OPPOSITION FILED WITHIN TIME LIMITSTAA | STAA | EP | |
| Fr: translation filedET | ET | EP | |
| It: translation for a ep patent filedITF | ITF | EP | |
| It: translation for a ep patent filedITF | ITF | EP | |
| Corresponds to:REF | REF | EP | |
| Designated contracting statesAK | AK | EP | |
| (expected) grantORIGINAL CODE: 0009210GRAA | GRAA | EP | |
| First examination report despatched17Q | 17Q | EP | |
| Request for examination filed17P | 17P | EP | |
| Designated contracting statesAK | AK | EP | |
| Search report despatchedORIGINAL CODE: 0009013PUAL | PUAL | EP | |
| Designated contracting statesAK | AK | EP | |
| Public reference made under article 153(3) epc to a published international application that has entered the european phaseORIGINAL CODE: 0009012PUAI | PUAI | EP |
Numbers
- Publication
- 0248634
- Publication, DOCDB
- 0248634
- Publication, EPODOC
- EP0248634
- Application
- 87304860
- Application, DOCDB
- 87304860
- Application, EPODOC
- EP19870304860
Titles3
- English
- Stabilized benzimidazole derivative and composition
- French
- Dérivé stabilisé de benzimidazole et composition
- German
- Stabilisiertes Benzimidazol-Derivat und Zusammenstellung
Classification
- CPC, 1
- C07D235/28
- IPC, 1
- C07D235 28
Designated states1
- Contracting states, 1
- Sweden