Nova Patents
ATE348809T1

Imides as inhibitors of TNF alpha

Abstract

A process of preparing thalidomide in which N-phthaloylglutamine or N-phthaloylisoglutamine is cyclized with N,N'-carbonyldiimidazole, characterised in that the process comprises heating said N-phthaloylglutamine or N-phthaloylisoglutamine and N,N'-carbonyldiimidazole in refluxing anhydrous tetrahydrofuran.

Term

Term ended

Projected expiry passed 1 July 2014, 12.2 years ago.

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84 members in 20 offices

This recordMember, by publication datePriority claim10 more offices are in the list below

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Priority claims
DocumentOfficeKindDate
8751093United States of AmericaA

Members84

Family members, oldest first
DocumentOfficeKind
CA2166315A1CanadaA1
CA2531868A1CanadaA1
CA2626178A1CanadaA1
WO9501348A2World Intellectual Property Organization (WIPO)A2
AU7216794AAustraliaA
WO9501348A3World Intellectual Property Organization (WIPO)A3
US5463063AUnited States of AmericaA
FI956362AFinlandA
FI956362LFinlandL
HU9600003D0HungaryD0
PL312386A1PolandA1
EP0706521A1European Patent Office (EPO)A1
KR960703891ARepublic of KoreaA
CZ1096A3CzechiaA3
SK166595A3SlovakiaA3
JPH09500872AJapanA
US5605914AUnited States of AmericaA
HUT75312AHungaryA
US5698579AUnited States of AmericaA
AU687843B2AustraliaB2
NZ268812ANew ZealandA
NZ329259ANew ZealandA
US5877200AUnited States of AmericaA
NZ329258ANew ZealandA
EP1004572A2European Patent Office (EPO)A2
EP1004580A2European Patent Office (EPO)A2
EP1004581A2European Patent Office (EPO)A2
US6075041AUnited States of AmericaA
HK1025765A1Hong Kong, ChinaA1
HK1025769A1Hong Kong, ChinaA1
PL180377B1PolandB1
US6200987B1United States of AmericaB1
RU2174516C2Russian FederationC2
EP1004581A3European Patent Office (EPO)A3
EP0706521B1European Patent Office (EPO)B1
EP1004572A3European Patent Office (EPO)A3
EP1004580A3European Patent Office (EPO)A3
AT225344TAustriaT
ATE225344T1AustriaT1
DE69431480D1GermanyD1
DK0706521T3DenmarkT3
PT706521EPortugalE
ES2184765T3SpainT3
HK1025770A1Hong Kong, ChinaA1
DE69431480T2GermanyT2
FI20040593AFinlandA
FI20040593A7FinlandA7
EP1004581B1European Patent Office (EPO)B1
AT277036TAustriaT
ATE277036T1AustriaT1
DE69434029D1GermanyD1
EP1477486A2European Patent Office (EPO)A2
EP1477486A3European Patent Office (EPO)A3
CZ294444B6CzechiaB6
DK1004581T3DenmarkT3
PT1004581EPortugalE
FI114984BFinlandB
ES2226696T3SpainT3
DE69434029T2GermanyT2
KR100401290B1Republic of KoreaB1
EP1004572B1European Patent Office (EPO)B1
AT319678TAustriaT
ATE319678T1AustriaT1
CA2166315CCanadaC
DE69434645D1GermanyD1
JP2006131647AJapanA
JP2006169261AJapanA
PT1004572EPortugalE
DK1004572T3DenmarkT3
JP2006188529AJapanA
JP2006188530AJapanA
ES2258956T3SpainT3
DE69434645T2GermanyT2
EP1004580B1European Patent Office (EPO)B1
AT348809TAustriaT
ATE348809T1This recordAustriaT1
DE69434895D1GermanyD1
PT1004580EPortugalE
DK1004580T3DenmarkT3
DE69434895T2GermanyT2
ES2278574T3SpainT3
JP3971794B2JapanB2
JP4461107B2JapanB2
CA2531868CCanadaC