PL370992A1
Inhibitors of histone deacetylase
Abstract
This invention comprises the novel compounds of formula (I) wherein n, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
Term
Term ended
Projected expiry passed 11 March 2023, 3.5 years ago.
- Priority
- Filed
- Published
- Projected expiry
- Today
287 members in 27 offices
Priority claims4
| Document | Office | Kind | Date |
|---|---|---|---|
| 36379902 | United States of America | P | |
| 36379902 | United States of America | P | |
| 0260363799 | – | – | – |
| US20020363799P | – | – | – |
Members287
| Document | Office | Kind | |
|---|---|---|---|
| CA2475764A1 | Canada | A1 | |
| CA2475766A1 | Canada | A1 | |
| CA2476065A1 | Canada | A1 | |
| CA2476067A1 | Canada | A1 | |
| CA2476186A1 | Canada | A1 | |
| CA2476296A1 | Canada | A1 | |
| CA2476583A1 | Canada | A1 | |
| CA2476586A1 | Canada | A1 | |
| WO03075929A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076395A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076400A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076401A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076421A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076422A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076430A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO03076438A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU2003209727A1 | Australia | A1 | |
| AU2003212335A1 | Australia | A1 | |
| AU2003212336A1 | Australia | A1 | |
| AU2003212337A1 | Australia | A1 | |
| AU2003218735A1 | Australia | A1 | |
| AU2003218736A1 | Australia | A1 | |
| AU2003218737A1 | Australia | A1 | |
| AU2003218738A1 | Australia | A1 | |
| TW200400822A | Taiwan Province of China | A | |
| TW200400941A | Taiwan Province of China | A | |
| TW200400961A | Taiwan Province of China | A | |
| TW200404794A | Taiwan Province of China | A | |
| TW200406382A | Taiwan Province of China | A | |
| NO20044113L | Norway | L | |
| NO20044135L | Norway | L | |
| NO20044146L | Norway | L | |
| NO20044194L | Norway | L | |
| NO20044224L | Norway | L | |
| NO20044314L | Norway | L | |
| MXPA04007775A | Mexico | A | |
| MXPA04007776A | Mexico | A | |
| KR20040090978A | Republic of Korea | A | |
| KR20040090979A | Republic of Korea | A | |
| KR20040090981A | Republic of Korea | A | |
| KR20040090985A | Republic of Korea | A | |
| KR20040093692A | Republic of Korea | A | |
| KR20040094672A | Republic of Korea | A | |
| MXPA04008795A | Mexico | A | |
| MXPA04008796A | Mexico | A | |
| MXPA04008797A | Mexico | A | |
| MXPA04008806A | Mexico | A | |
| EP1485099A1 | European Patent Office (EPO) | A1 | |
| EP1485348A1 | European Patent Office (EPO) | A1 | |
| EP1485353A1 | European Patent Office (EPO) | A1 | |
| EP1485354A1 | European Patent Office (EPO) | A1 | |
| EP1485364A1 | European Patent Office (EPO) | A1 | |
| EP1485365A1 | European Patent Office (EPO) | A1 | |
| EP1485370A1 | European Patent Office (EPO) | A1 | |
| EP1485378A1 | European Patent Office (EPO) | A1 | |
| BR0307575A | Brazil | A | |
| BR0307606A | Brazil | A | |
| BR0307607A | Brazil | A | |
| BR0308081A | Brazil | A | |
| BR0307624A | Brazil | A | |
| BR0307599A | Brazil | A | |
| AR039564A1 | Argentina | A1 | |
| AR039565A1 | Argentina | A1 | |
| AR039566A1 | Argentina | A1 | |
| AR039567A1 | Argentina | A1 | |
| AR039568A1 | Argentina | A1 | |
| EA200401197A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200401199A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200401200A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200401201A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200401202A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EA200401204A1 | Eurasian Patent Organization (EAPO) | A1 | |
| HRP20040803A2 | Croatia | A2 | |
| HRP20040804A2 | Croatia | A2 | |
| HRP20040799A2 | Croatia | A2 | |
| HRP20040801A2 | Croatia | A2 | |
| HRP20040805A2 | Croatia | A2 | |
| US2005096468A1 | United States of America | A1 | |
| US2005107384A1 | United States of America | A1 | |
| US2005113373A1 | United States of America | A1 | |
| US2005119250A1 | United States of America | A1 | |
| PL370982A1 | Poland | A1 | |
| PL370990A1 | Poland | A1 | |
| PL370991A1 | Poland | A1 | |
| PL370992A1This record | Poland | A1 | |
| PL371036A1 | Poland | A1 | |
| PL371100A1 | Poland | A1 | |
| HRP20040802A2 | Croatia | A2 | |
| JP2005519950A | Japan | A | |
| US2005148613A1 | United States of America | A1 | |
| CN1639125A | China | A | |
| CN1642551A | China | A | |
| CN1642907A | China | A | |
| CN1642912A | China | A | |
| CN1642931A | China | A | |
| CN1642948A | China | A | |
| US2005165016A1 | United States of America | A1 | |
| NZ534834A | New Zealand | A | |
| US2005171347A1 | United States of America | A1 | |
| JP2005523907A | Japan | A |
Showing 100 of 287
Numbers
- Publication, DOCDB
- 370992
- Publication, EPODOC
- PL370992
- Application
- 3370992
- Application, DOCDB
- 37099203
- Application, EPODOC
- PL20030370992
Titles2
- English
- INHIBITORS OF HISTONE DEACETYLASE
- Polish
- Inhibitory deacetylazy histonowej
Classification
- CPC, 76
- C07D295/26
- C07D413/12
- C07D207/09
- C07D207/14
- C07D211/58
- C07D213/78
- C07D217/02
- C07D239/42
- C07D295/155
- C07D307/68
- C07D401/04
- C07D403/04
- C07D409/12
- C07D413/04
- C07D471/04
- C07D471/10
- C07D513/04
- C12Q1/48
- C07D401/12
- C07D211/14
- C07D217/04
- A61K31/402
- C07D409/14
- A61K31/4545
- C07D403/12
- C12Q1/34
- A61K31/40
- A61K31/472
- A61K31/496
- C07D217/16
- C07D405/06
- A61K31/435
- A61K31/495
- A61K31/506
- A61K45/06
- A61K31/4427
- A61K31/454
- A61K31/5377
- A61K31/55
- A61P1/04
- A61P11/00
- A61P11/02
- A61P11/06
- A61P13/08
- A61P13/10
- A61P13/12
- A61P15/00
- A61P17/00
- A61P17/04
- A61P17/06
- A61P17/10
- A61P17/14
- A61P17/16
- A61P19/02
- A61P19/06
- A61P21/04
- A61P25/00
- A61P25/16
- A61P25/28
- A61P27/02
- A61P27/06
- A61P29/00
- A61P3/10
- A61P31/18
- A61P35/00
- A61P35/02
- A61P37/02
- A61P37/04
- A61P37/06
- A61P37/08
- A61P43/00
- A61P5/00
- A61P9/00
- A61P9/02
- A61P9/08
- A61P9/10
- IPC, 85
- A61K31 40
- A61K31 438
- C07D249 12
- A61K31 4427
- A61K31 445
- A61K31 4545
- A61K31 472
- A61K31 495
- A61K31 496
- A61K31 497
- A61K31 506
- A61K31 517
- A61K31 53
- A61K31 5377
- A61K31 55
- A61K31 551
- A61K45 00
- A61P1 04
- A61P3 10
- A61P5 00
- A61P9 00
- A61P9 02
- A61P9 08
- A61P9 10
- A61P11 00
- A61P11 02
- A61P11 06
- A61P13 08
- A61P13 10
- A61P13 12
- A61P15 00
- A61P17 00
- A61P17 04
- A61P17 06
- A61P17 10
- A61P17 14
- A61P17 16
- A61P19 02
- A61P19 06
- A61P21 04
- A61P25 00
- A61P25 16
- A61P25 28
- A61P27 02
- A61P27 06
- A61P29 00
- A61P31 18
- A61P35 00
- A61P35 02
- A61P37 02
- A61P37 04
- A61P37 06
- A61P37 08
- A61P43 00
- C07D207 09
- C07D207 14
- C07D211 26
- C07D211 58
- C07D213 74
- C07D213 78
- C07D217 02
- C07D217 04
- C07D239 42
- C07D241 04
- C07D295 14
- C07D295 155
- C07D295 20
- C07D295 22
- C07D295 26
- C07D307 68
- C07D317 58
- C07D401 04
- C07D401 06
- C07D401 12
- C07D401 14
- C07D403 04
- C07D403 12
- C07D405 12
- C07D405 14
- C07D409 12
- C07D413 02
- C07D413 04
- C07D413 12
- C07D471 10
- C12Q1 48