Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof
Abstract
The present invention relates generally to the field of ligands for nicotinic acetylcholine receptors (nAChR), activation of nAChRs, and treatment of disease states associated with defective or malfunctioning nicotinic acetylcholine receptors, particularly in the brain. Furthermore, the invention relates to novel compounds (indazoles and benzothiazoles) which act as ligands for the α7-nAChRound type, methods of preparing such compounds, compositions containing such compounds, and methods of use thereof.
Term
No projected expiry on record.
- Priority
- Filed
- Published
- Today
1 claim: 1 independent, 0 dependent
- 1Den foreliggende oppfinnelse vedrører generelt området ligander for nikotinacetylkolinreseptorer (nAChR), aktivering av nAChR-er og behandling av sykdomstilstander forbundet med defekte eller dårlig virkende nikotinacetylkolinreseptorer, spesielt i hjernen. Videre vedrører oppfinnelsen nye forbindelser (indazoler og benzotiazoler) som virker som ligander for a7-nAChRundertypen, fremgangsmåter for fremstilling av slike forbindelser, preparater som inneholder slike forbindelser, og fremgangsmåter for anvendelse derav.
4 paragraphs, as filed
Brian Herbert, 3 Grandview Avenue, NJ07460 STOCKHOLM, US
True Minh Nguyen, 3 East 101st Street, Apt 5E, NY10029 NEW YORK, US Wenge Xie, 2347 Pembroke Court, NJ07430 MAHWAH, US Carla Maria Gauss, 4 Washington Square Village, Apt 5P, NY10012 NEW YORK, US Tandberg Patent Office AS,
PO Box 7085 Majorstua, 0306 OSLO, NO (74) Proxy (54) Name Indazoles, benzothiazoles and benzoisothiazoles, and their manufacture and uses.
(57) Summary
49 members in 25 offices
Priority claims12
| Document | Office | Kind | Date |
|---|---|---|---|
| 41315102 | United States of America | P | |
| 41315102 | United States of America | P | |
| 44846903 | United States of America | P | |
| 44846903 | United States of America | P | |
| 0329976 | United States of America | W | |
| 0329976 | United States of America | W | |
| 413151 | – | – | – |
| 448469 | – | – | – |
| PCTUS0329976 | – | – | – |
| US20020413151P | – | – | – |
| US20030448469P | – | – | – |
| WO2003US29976 | – | – | – |
Members49
| Document | Office | Kind | |
|---|---|---|---|
| CA2499128A1 | Canada | A1 | |
| WO2004029050A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU2003276919A1 | Australia | A1 | |
| US2004132790A1 | United States of America | A1 | |
| NO20051985LThis record | Norway | L | |
| EE200500011A | Estonia | A | |
| EP1543000A1 | European Patent Office (EPO) | A1 | |
| MA27453A1 | Morocco | A1 | |
| KR20050069999A | Republic of Korea | A | |
| MXPA05003317A | Mexico | A | |
| BR0314485A | Brazil | A | |
| SK50322005A3 | Slovakia | A3 | |
| CN1684962A | China | A | |
| HRP20050266A2 | Croatia | A2 | |
| CZ2005252A3 | Czechia | A3 | |
| HUP0500610A2 | Hungary | A2 | |
| PL375764A1 | Poland | A1 | |
| BG109117A | Bulgaria | A | |
| ZA200502465B | South Africa | B | |
| JP2006503851A | Japan | A | |
| RU2005112712A | Russian Federation | A | |
| HK1083831A | Hong Kong, China | A | |
| NZ539049A | New Zealand | A | |
| RS20050248A | Serbia | A | |
| US2008154037A1 | United States of America | A1 | |
| US2008176890A1 | United States of America | A1 | |
| US7429664B2 | United States of America | B2 | |
| CN100484937C | China | C | |
| US2009209579A1 | United States of America | A1 | |
| RU2391341C2 | Russian Federation | C2 | |
| EP2305675A1 | European Patent Office (EPO) | A1 | |
| US7943773B2 | United States of America | B2 | |
| JP2011140509A | Japan | A | |
| US2011212957A1 | United States of America | A1 | |
| PL210065B1 | Poland | B1 | |
| EE05516B1 | Estonia | B1 | |
| JP4890762B2 | Japan | B2 | |
| US8134003B2 | United States of America | B2 | |
| KR101129933B1 | Republic of Korea | B1 | |
| US2012101094A1 | United States of America | A1 | |
| CA2499128C | Canada | C | |
| US8252811B2 | United States of America | B2 | |
| NO332535B1 | Norway | B1 | |
| EP1543000B1 | European Patent Office (EPO) | B1 | |
| AU2003276919B2 | Australia | B2 | |
| ES2405594T3 | Spain | T3 | |
| SK288115B6 | Slovakia | B6 | |
| HUP0500610A3 | Hungary | A3 | |
| RS53147B | Serbia | B |
1 legal event, as the office reported them to INPADOC
Events
| Event | Code | |
|---|---|---|
| Lapsed by not paying the annual feesLapsedMM1K | MM1K |
Numbers
- Publication, DOCDB
- 20051985
- Publication, EPODOC
- NO20051985L
- Application
- 1985
- Application, DOCDB
- 20051985
- Application, EPODOC
- NO20050001985
Titles2
- Norwegian
- Indazoler, benzotiazoler og benzoisotiazoler, samt fremstilling og anvendelser derav.
- English
- Indazoles, benzothiazoles and benzoisothiazoles, and their preparation and uses.
Classification
- CPC, 25
- C07D453/02
- A61P23/00
- A61P25/00
- A61P25/04
- A61P25/06
- A61P25/08
- A61P25/14
- A61P25/16
- A61P25/18
- A61P25/20
- A61P25/22
- A61P25/24
- A61P25/28
- A61P25/32
- A61P25/34
- A61P29/00
- A61P3/04
- A61P31/18
- A61P39/00
- A61P41/00
- A61P43/00
- A61P9/00
- A61P9/10
- A61P3/10
- A61K31/439
- IPC, 2
- A61P25 28
- C07D453 02