BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF IgE
Abstract
The present invention is directed to small molecule inhibitors of the IgE response to allergens which are useful in the treatment of allergy and/or asthma or any diseases where IgE is pathogenic.
Term
No projected expiry on record.
- Priority
- Filed
- Published
- Today
1 claim: 1 independent, 0 dependent
- 1Michael W Major, San Diego, CA, US Bryns Zacco AS, 0106 Oslo Forbindelser med IgE-påvirkende egenskaper Småmolekyl-inhibitorer av IgE-responsen til allergener som er nyttige i behandlingen av allergi og/eller astma eller hvilke som helst sykdommer hvor IgE er patogent.
9 paragraphs, as filed
(22) On day (24) Running day (41) Alm. avail.
(71) Seeking (72) Inventor (74) Proxy (54) Title (57) Summary
<td>20005887 2000.11.21</td><td>(86) Int. Entry day and search number</td><td>1999.05.21, PCT / US99 / 11363</td>
<td>1999.05.21</td><td>(85) Date of transfer</td><td>2000,11.21</td>
<td>2001.01.19</td><td>(30) Priority</td><td>1998.05.22, US, 86494</td>
Avanir Pharmaceuticals, 1388 Sorrento Valley Road, San Diego, CA 92121, US
Jagadish Sircar, San Diego, CA, US
Mark L Richards, San Diego, CA, US
Michael G Campbell, San Diego, CA, US
119 members in 26 offices
Priority claims8
| Document | Office | Kind | Date |
|---|---|---|---|
| 8649498 | United States of America | P | |
| 8649498 | United States of America | P | |
| 9911363 | United States of America | W | |
| 9911363 | United States of America | W | |
| 8649498 | – | – | – |
| 9911363 | – | – | – |
| US19980086494P | – | – | – |
| WO1999US11363 | – | – | – |
Members119
| Document | Office | Kind | |
|---|---|---|---|
| CA2332985A1 | Canada | A1 | |
| CA2332989A1 | Canada | A1 | |
| CA2332999A1 | Canada | A1 | |
| WO9961013A2 | World Intellectual Property Organization (WIPO) | A2 | |
| WO9961019A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO9961020A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU4094299A | Australia | A | |
| AU4197899A | Australia | A | |
| AU4312099A | Australia | A | |
| WO9961013A3 | World Intellectual Property Organization (WIPO) | A3 | |
| NO20005887D0 | Norway | D0 | |
| NO20005888D0 | Norway | D0 | |
| NO20005889D0 | Norway | D0 | |
| NO20005887LThis record | Norway | L | |
| NO20005888L | Norway | L | |
| NO20005889L | Norway | L | |
| EP1077695A2 | European Patent Office (EPO) | A2 | |
| EP1077700A1 | European Patent Office (EPO) | A1 | |
| EP1079830A1 | European Patent Office (EPO) | A1 | |
| KR20010030179A | Republic of Korea | A | |
| ZA200007753B | South Africa | B | |
| US6271390B1 | United States of America | B1 | |
| ZA200007754B | South Africa | B | |
| CN1311675A | China | A | |
| CN1311679A | China | A | |
| BR9910641A | Brazil | A | |
| BR9910642A | Brazil | A | |
| US6303645B1 | United States of America | B1 | |
| CN1317965A | China | A | |
| CZ20004351A3 | Czechia | A3 | |
| HU0102550A2 | Hungary | A2 | |
| HUP0102550A2 | Hungary | A2 | |
| BR9910640A | Brazil | A | |
| HK1035326A1 | Hong Kong, China | A1 | |
| PL345219A1 | Poland | A1 | |
| ZA200007752B | South Africa | B | |
| PL345560A1 | Poland | A1 | |
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| HUP0101894A2 | Hungary | A2 | |
| HU0102128A2 | Hungary | A2 | |
| HUP0102128A2 | Hungary | A2 | |
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| HUP0102128A3 | Hungary | A3 | |
| JP2002516274A | Japan | A | |
| JP2002516276A | Japan | A | |
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| US6451829B2 | United States of America | B2 | |
| CA2441177A1 | Canada | A1 | |
| US2002132808A1 | United States of America | A1 | |
| WO02072090A1 | World Intellectual Property Organization (WIPO) | A1 | |
| MXPA00011467A | Mexico | A | |
| MXPA00011470A | Mexico | A | |
| AU754562B2 | Australia | B2 | |
| AU754943B2 | Australia | B2 | |
| HU0102550A3 | Hungary | A3 | |
| HUP0102550A3 | Hungary | A3 | |
| MXPA00011422A | Mexico | A | |
| US2003004203A1 | United States of America | A1 | |
| US2003100582A1 | United States of America | A1 | |
| NZ508413A | New Zealand | A | |
| EP1368028A1 | European Patent Office (EPO) | A1 | |
| AR034023A1 | Argentina | A1 | |
| NZ508416A | New Zealand | A | |
| HU0303460A2 | Hungary | A2 | |
| HUP0303460A2 | Hungary | A2 | |
| KR20040025903A | Republic of Korea | A | |
| IL157730D0 | Israel | D0 | |
| CZ20032691A3 | Czechia | A3 | |
| MXJL03000027A | Mexico | A | |
| CN1496257A | China | A | |
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| UA67774C2 | Ukraine | C2 | |
| UA67775C2 | Ukraine | C2 | |
| HU0303460A3 | Hungary | A3 | |
| HUP0303460A3 | Hungary | A3 | |
| ZA200307916B | South Africa | B | |
| JP2004528304A | Japan | A | |
| RU2236220C2 | Russian Federation | C2 | |
| RU2236221C2 | Russian Federation | C2 | |
| US2004214821A1 | United States of America | A1 | |
| PL364230A1 | Poland | A1 | |
| BR0208010A | Brazil | A | |
| RU2003127367A | Russian Federation | A | |
| EP1077700B1 | European Patent Office (EPO) | B1 | |
| US2005075343A1 | United States of America | A1 | |
| AT292465T | Austria | T | |
| ATE292465T1 | Austria | T1 | |
| DE69924607D1 | Germany | D1 | |
| NZ528835A | New Zealand | A | |
| US6911462B2 | United States of America | B2 | |
| US6919366B2 | United States of America | B2 |
1 legal event, as the office reported them to INPADOC
Events
| Event | Code | |
|---|---|---|
| Withdrawal, rejection or dismissal of laid open patent applicationFC2A | FC2A |
Numbers
- Publication, DOCDB
- 20005887
- Publication, EPODOC
- NO20005887L
- Application
- 5887
- Application, DOCDB
- 20005887
- Application, EPODOC
- NO20000005887
Titles2
- English
- Compounds with IgE-affecting properties
- Norwegian
- Forbindelser med IgE-påvirkende egenskaper
Classification
- CPC, 9
- A61K31/415
- A61K31/00
- A61K31/4184
- A61K31/4545
- A61K45/06
- A61P11/06
- A61P37/00
- A61P37/08
- A61P43/00
- IPC, 47
- A61K31 00
- A61K31 166
- A61K31 167
- C07D235 14
- A61K31 18
- A61K31 337
- A61K31 357
- A61K31 382
- A61K31 397
- A61K31 403
- A61K31 4035
- A61K31 404
- A61K31 4045
- A61K31 415
- A61K31 4184
- A61K31 42
- A61K31 423
- A61K31 4427
- A61K31 443
- A61K31 4433
- A61K31 4439
- A61K31 445
- A61K31 451
- A61K31 454
- A61K31 4545
- A61K31 53
- A61K45 06
- A61P11 06
- A61P37 08
- A61P43 00
- C07D205 04
- C07D209 16
- C07D209 48
- C07D211 46
- C07D211 52
- C07D235 18
- C07D251 70
- C07D261 12
- C07D319 18
- C07D401 12
- C07D401 14
- C07D403 14
- C07D405 04
- C07D405 12
- C07D409 12
- C07D409 14
- C07D413 04