MD20140004A2
Deuterated 1-piperazino-3-phenyl-indanes for treatment of schizophrenia
Abstract
The present invention relates to deuterated 1-piperazino-3-phenyl-indanes and salts thereof with activity at dopamine receptors D1 and D2 as well as the 5HT2 receptors in the central nervous system, to medicaments comprising such compounds as active ingredients, to the use of such compounds in the treatment of diseases in the central nervous system, and to methods of treatment comprising administration of such compounds.
Term
No projected expiry on record.
- Priority
- Filed
- Published
- Today
139 members in 47 offices
Priority claims12
| Document | Office | Kind | Date |
|---|---|---|---|
| 201161498651 | United States of America | P | |
| 201161498651 | United States of America | P | |
| 201161537103 | United States of America | P | |
| 201161537103 | United States of America | P | |
| 2012001386 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| 2012001386 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| 61498651 | – | – | – |
| 61537103 | – | – | – |
| PCTIB12001386 | – | – | – |
| US201161498651P | – | – | – |
| US201161537103P | – | – | – |
| WO2012IB01386 | – | – | – |
Members139
| Document | Office | Kind | |
|---|---|---|---|
| US2012322811A1 | United States of America | A1 | |
| CA2837820A1 | Canada | A1 | |
| WO2012176066A1 | World Intellectual Property Organization (WIPO) | A1 | |
| TW201311248A | Taiwan Province of China | A | |
| WO2013043373A1 | World Intellectual Property Organization (WIPO) | A1 | |
| US2013281436A1 | United States of America | A1 | |
| US8575174B2 | United States of America | B2 | |
| AU2012273657A1 | Australia | A1 | |
| AP2013007338A0 | African Regional Intellectual Property Organization (ARIPO) | A0 | |
| CO6821965A2 | Colombia | A2 | |
| IL229640A0 | Israel | A0 | |
| IL229640D0 | Israel | D0 | |
| AR086987A1 | Argentina | A1 | |
| PH12013502598A1 | Philippines | A1 | |
| DOP2013000305A | Dominican Republic | A | |
| ECSP14013155A | Ecuador | A | |
| CN103649019A | China | A | |
| CR20130654A | Costa Rica | A | |
| MX2013014849A | Mexico | A | |
| KR20140041567A | Republic of Korea | A | |
| EP2720989A1 | European Patent Office (EPO) | A1 | |
| CN103765044A | China | A | |
| DE112012003408T5 | Germany | T5 | |
| KR20140065437A | Republic of Korea | A | |
| MD20140004A2This record | Republic of Moldova | A2 | |
| MA35268B1 | Morocco | B1 | |
| US2014187367A1 | United States of America | A1 | |
| US2014187368A1 | United States of America | A1 | |
| US2014187369A1 | United States of America | A1 | |
| CL2013003646A1 | Chile | A1 | |
| EA201490045A1 | Eurasian Patent Organization (EAPO) | A1 | |
| JP2014520140A | Japan | A | |
| WO2014137790A1 | World Intellectual Property Organization (WIPO) | A1 | |
| PE20141113A1 | Peru | A1 | |
| JP2014528047A | Japan | A | |
| HK1197228A | Hong Kong, China | A | |
| HK1197228A1 | Hong Kong, China | A1 | |
| GT201300304A | Guatemala | A | |
| JP5668177B2 | Japan | B2 | |
| ZA201309613B | South Africa | B | |
| NZ618222A | New Zealand | A | |
| TN2013000503A1 | Tunisia | A1 | |
| US9012453B2 | United States of America | B2 | |
| PE20150928A1 | Peru | A1 | |
| AP3310A | African Regional Intellectual Property Organization (ARIPO) | A | |
| CN103649019B | China | B | |
| DE112014000738T5 | Germany | T5 | |
| RU2014113136A | Russian Federation | A | |
| US2015307458A1 | United States of America | A1 | |
| CN105102859A | China | A | |
| KR20150141183A | Republic of Korea | A | |
| US9216961B2 | United States of America | B2 | |
| UA110526C2 | Ukraine | C2 | |
| US2016068497A1 | United States of America | A1 | |
| JP2016509185A | Japan | A | |
| MX339552B | Mexico | B | |
| US9360088B2 | United States of America | B2 | |
| US9377087B2 | United States of America | B2 | |
| US9377088B2 | United States of America | B2 | |
| AU2012273657B2 | Australia | B2 | |
| EP2720989B1 | European Patent Office (EPO) | B1 | |
| US2016245375A1 | United States of America | A1 | |
| US2016245376A1 | United States of America | A1 | |
| EA024651B1 | Eurasian Patent Organization (EAPO) | B1 | |
| PT2720989T | Portugal | T | |
| LT2720989T | Lithuania | T | |
| DK2720989T3 | Denmark | T3 | |
| SI2720989T1 | Slovenia | T1 | |
| HRP20161348T1 | Croatia | T1 | |
| BR112013031702A2 | Brazil | A2 | |
| SMT201600383B | San Marino | B | |
| CN103765044B | China | B | |
| ES2601213T3 | Spain | T3 | |
| ME02513B | Montenegro | B | |
| EP3135656A1 | European Patent Office (EPO) | A1 | |
| RS55304B1 | Serbia | B1 | |
| US9617231B2 | United States of America | B2 | |
| GEP201706655B | Georgia | B | |
| PL2720989T3 | Poland | T3 | |
| US2017158650A1 | United States of America | A1 | |
| CY1118158T1 | Cyprus | T1 | |
| HUE030883T2 | Hungary | T2 | |
| TW201722895A | Taiwan Province of China | A | |
| JP6189846B2 | Japan | B2 | |
| JO3128B1 | Jordan | B1 | |
| CN105102859B | China | B | |
| JP2017215046A | Japan | A | |
| MD4538B1 | Republic of Moldova | B1 | |
| US9879764B2 | United States of America | B2 | |
| TWI614234B | Taiwan Province of China | B | |
| IL229640A | Israel | A | |
| IL229640B | Israel | B | |
| US2018112748A1 | United States of America | A1 | |
| TWI627956B | Taiwan Province of China | B | |
| KR20180075717A | Republic of Korea | A | |
| KR101879474B1 | Republic of Korea | B1 | |
| JP6359571B2 | Japan | B2 | |
| MY166773A | Malaysia | A | |
| MD4538C1 | Republic of Moldova | C1 | |
| US10118907B2 | United States of America | B2 |
Showing 100 of 139
1 legal event, as the office reported them to INPADOC
Events
| Event | Code | |
|---|---|---|
| Patent for invention issuedFG4A | FG4A |
Numbers
- Publication
- 0020140004
- Publication, DOCDB
- 20140004
- Publication, EPODOC
- MD20140004
- Application
- 20140004
- Application, DOCDB
- 20140004
- Application, EPODOC
- MD20140000004
Titles3
- English
- Deuterated 1-piperazino-3-phenyl-indanes for treatment of schizophrenia
- Romanian
- 1-Piperazino-3-fenil-indani deuteraţi pentru tratamentul schizofreniei
- Russian
- Дейтерированные 1-пиперазино-3-фенилинданы для лечения шизофрении
Classification
- CPC, 18
- C07D241/04
- C07D295/073
- C07B59/002
- A61K31/451
- A61K31/454
- A61K31/4545
- A61K31/495
- A61K31/496
- A61K31/519
- A61K31/551
- A61K31/554
- A61P25/00
- A61P25/18
- A61P25/24
- A61P25/28
- C07C45/61
- C07C45/67
- C07B2200/05
- IPC, 4
- C07B59 00
- A61K31 495
- A61P25 00
- C07D241 04