MA28629B1
Benzothiazepine derivatives as ryanodine receptor (RYR2) inhibitors and their use in the treatment of cardiac diseases
Abstract
The present application relates to benzothiazepine S36 and its oxidized derivatives tor use in limiting or preventing a decrease in the level of RyR2-bound FKBP12.6 in a subject having a cardiac condition or in treating or preventing a cardiac condition in a subject.
Term
No projected expiry on record.
- Priority
- Filed
- Granted
- Today
210 members in 37 offices
Priority claims4
| Document | Office | Kind | Date |
|---|---|---|---|
| 80908904 | United States of America | A | |
| 80908904 | United States of America | A | |
| 10809089 | – | – | – |
| US20040809089 | – | – | – |
Members210
| Document | Office | Kind | |
|---|---|---|---|
| US6489125B1 | United States of America | B1 | |
| US2003134331A1 | United States of America | A1 | |
| US2004048780A1 | United States of America | A1 | |
| AU2004220548A1 | Australia | A1 | |
| WO2004080283A2 | World Intellectual Property Organization (WIPO) | A2 | |
| US2004224368A1 | United States of America | A1 | |
| US2004229781A1 | United States of America | A1 | |
| AU2004253523A1 | Australia | A1 | |
| CA2530594A1 | Canada | A1 | |
| WO2005002518A2 | World Intellectual Property Organization (WIPO) | A2 | |
| AU2004281672A1 | Australia | A1 | |
| CA2541847A1 | Canada | A1 | |
| WO2005037195A2 | World Intellectual Property Organization (WIPO) | A2 | |
| US2005186640A1 | United States of America | A1 | |
| US2005187386A1 | United States of America | A1 | |
| US2005215540A1 | United States of America | A1 | |
| AU2005227907A1 | Australia | A1 | |
| CA2560866A1 | Canada | A1 | |
| WO2005094457A2 | World Intellectual Property Organization (WIPO) | A2 | |
| WO2005002518A3 | World Intellectual Property Organization (WIPO) | A3 | |
| WO2005037195A3 | World Intellectual Property Organization (WIPO) | A3 | |
| EP1603450A2 | European Patent Office (EPO) | A2 | |
| EP1635801A2 | European Patent Office (EPO) | A2 | |
| MXPA06000138A | Mexico | A | |
| WO2005094457A3 | World Intellectual Property Organization (WIPO) | A3 | |
| WO2005094457B1 | World Intellectual Property Organization (WIPO) | B1 | |
| CA2591924A1 | Canada | A1 | |
| WO2006071603A2 | World Intellectual Property Organization (WIPO) | A2 | |
| NO20062063L | Norway | L | |
| EP1684735A2 | European Patent Office (EPO) | A2 | |
| US2006194767A1 | United States of America | A1 | |
| MA28146A1 | Morocco | A1 | |
| AU2005329398A1 | Australia | A1 | |
| AU2005329399A1 | Australia | A1 | |
| CA2601541A1 | Canada | A1 | |
| WO2006101496A1 | World Intellectual Property Organization (WIPO) | A1 | |
| WO2006101497A2 | World Intellectual Property Organization (WIPO) | A2 | |
| WO2006071603A3 | World Intellectual Property Organization (WIPO) | A3 | |
| KR20060110290A | Republic of Korea | A | |
| EA200600740A1 | Eurasian Patent Organization (EAPO) | A1 | |
| BRPI0415434A | Brazil | A | |
| NO20064843L | Norway | L | |
| CN1886122A | China | A | |
| EP1734969A2 | European Patent Office (EPO) | A2 | |
| US2006293266A1 | United States of America | A1 | |
| AU2006283534A1 | Australia | A1 | |
| CA2620183A1 | Canada | A1 | |
| US2007049572A1 | United States of America | A1 | |
| WO2007024717A2 | World Intellectual Property Organization (WIPO) | A2 | |
| JP2007507536A | Japan | A | |
| WO2006071603A9 | World Intellectual Property Organization (WIPO) | A9 | |
| KR20070041432A | Republic of Korea | A | |
| MA28629B1This record | Morocco | B1 | |
| CN1980677A | China | A | |
| US2007173482A1 | United States of America | A1 | |
| WO2006101497A3 | World Intellectual Property Organization (WIPO) | A3 | |
| BRPI0509199A | Brazil | A | |
| JP2007524631A | Japan | A | |
| JP2007525165A | Japan | A | |
| EA200601765A1 | Eurasian Patent Organization (EAPO) | A1 | |
| JP2007530561A | Japan | A | |
| WO2007127145A2 | World Intellectual Property Organization (WIPO) | A2 | |
| EP1861385A1 | European Patent Office (EPO) | A1 | |
| EP1861707A2 | European Patent Office (EPO) | A2 | |
| KR20070116900A | Republic of Korea | A | |
| MX2007011528A | Mexico | A | |
| WO2007143112A2 | World Intellectual Property Organization (WIPO) | A2 | |
| NO20075386L | Norway | L | |
| AR057776A1 | Argentina | A1 | |
| US7312044B2 | United States of America | B2 | |
| TW200800930A | Taiwan Province of China | A | |
| EP1635801A4 | European Patent Office (EPO) | A4 | |
| WO2008021432A2 | World Intellectual Property Organization (WIPO) | A2 | |
| WO2008021439A2 | World Intellectual Property Organization (WIPO) | A2 | |
| WO2007143112A3 | World Intellectual Property Organization (WIPO) | A3 | |
| CN101146785A | China | A | |
| TW200815381A | Taiwan Province of China | A | |
| EA200702057A1 | Eurasian Patent Organization (EAPO) | A1 | |
| KR20080037741A | Republic of Korea | A | |
| WO2008060332A2 | World Intellectual Property Organization (WIPO) | A2 | |
| NO20081421L | Norway | L | |
| WO2008064264A2 | World Intellectual Property Organization (WIPO) | A2 | |
| EP1928850A2 | European Patent Office (EPO) | A2 | |
| US7393652B2 | United States of America | B2 | |
| WO2008060332A9 | World Intellectual Property Organization (WIPO) | A9 | |
| AR060986A1 | Argentina | A1 | |
| ECSP088306A | Ecuador | A | |
| ZA200707573B | South Africa | B | |
| AR061173A1 | Argentina | A1 | |
| AR061174A1 | Argentina | A1 | |
| JP2008534497A | Japan | A | |
| EA200800665A1 | Eurasian Patent Organization (EAPO) | A1 | |
| MA29785B1 | Morocco | B1 | |
| WO2008060332A8 | World Intellectual Property Organization (WIPO) | A8 | |
| WO2007127145A3 | World Intellectual Property Organization (WIPO) | A3 | |
| WO2008021432A3 | World Intellectual Property Organization (WIPO) | A3 | |
| WO2004080283A3 | World Intellectual Property Organization (WIPO) | A3 | |
| WO2008021439A3 | World Intellectual Property Organization (WIPO) | A3 | |
| SG147414A1 | Singapore | A1 | |
| WO2008064264A8 | World Intellectual Property Organization (WIPO) | A8 |
Showing 100 of 210
Numbers
- Publication, DOCDB
- 28629
- Publication, EPODOC
- MA28629
- Application
- 29403
- Application, DOCDB
- 29403
- Application, EPODOC
- MA20060029403
Titles2
- French
- NOUVEAUX MEDICAMENTS ANTI-ARHYTHMIQUES CONTRE L'INFARCTUS CIBLANT LA FUITE DU RECEPTEUR DE RYANODINE (RYR2) ET LEURS UTILISATIONS
- English
- NOVEL ARTHRHYTHMIC DRUGS AGAINST INFARCTUS TARGETING RYANODINE RECEPTOR (RYR2) LEAKAGE AND USES THEREOF
Classification
- CPC, 6
- A61K31/554
- A61K31/553
- A61P43/00
- A61P9/00
- A61P9/04
- A61P9/06
- IPC, 1
- A61K31 554