IS7337A
Nicotinamide derivates useful as P38 inhibitors
Abstract
Compounds of formula (I): are inhibitors of p38 kinase and are useful in the treatment of conditions or disease states mediated by p38 kinase activity or mediated by cytokines produced by the activity of p38.
Term
Term ended
Projected expiry passed 28 June 2024, 2.2 years ago.
- Priority
- Filed and published
- Projected expiry
- Today
64 members in 27 offices
Priority claims11
| Document | Office | Kind | Date |
|---|---|---|---|
| 0203301 | United Kingdom | A | |
| 0203301 | United Kingdom | A | |
| 0225385 | United Kingdom | A | |
| 0225385 | United Kingdom | A | |
| 0300554 | United Kingdom | W | |
| 0300554 | United Kingdom | W | |
| GB02033017A | – | – | – |
| GB20020003301 | – | – | – |
| GB20020025385 | – | – | – |
| PCTGB0300554 | – | – | – |
| WO2003GB00554 | – | – | – |
Members64
| Document | Office | Kind | |
|---|---|---|---|
| GB0203301D0 | United Kingdom | D0 | |
| GB0225385D0 | United Kingdom | D0 | |
| CA2474192A1 | Canada | A1 | |
| WO03068747A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU2003207298A1 | Australia | A1 | |
| IS7337AThis record | Iceland | A | |
| NO20043176L | Norway | L | |
| KR20040082425A | Republic of Korea | A | |
| MXPA04007838A | Mexico | A | |
| EP1474395A1 | European Patent Office (EPO) | A1 | |
| BR0307351A | Brazil | A | |
| RU2004120553A | Russian Federation | A | |
| CN1633416A | China | A | |
| HK1070896A1 | Hong Kong, China | A1 | |
| JP2005519932A | Japan | A | |
| PL372628A1 | Poland | A1 | |
| US2005176964A1 | United States of America | A1 | |
| ZA200405602B | South Africa | B | |
| NZ533865A | New Zealand | A | |
| CO5611147A2 | Colombia | A2 | |
| US7125898B2 | United States of America | B2 | |
| US2006264479A1 | United States of America | A1 | |
| US2006276516A1 | United States of America | A1 | |
| EP1474395B1 | European Patent Office (EPO) | B1 | |
| RU2309951C2 | Russian Federation | C2 | |
| AT375980T | Austria | T | |
| DE60316913D1 | Germany | D1 | |
| EP1864975A2 | European Patent Office (EPO) | A2 | |
| PT1474395E | Portugal | E | |
| EP1864975A3 | European Patent Office (EPO) | A3 | |
| DK1474395T3 | Denmark | T3 | |
| CN100369898C | China | C | |
| SI1474395T1 | Slovenia | T1 | |
| ES2295553T3 | Spain | T3 | |
| HK1113056A1 | Hong Kong, China | A1 | |
| DE60316913T2 | Germany | T2 | |
| US7514456B2 | United States of America | B2 | |
| NO327418B1 | Norway | B1 | |
| IS2520B | Iceland | B | |
| AU2003207298B2 | Australia | B2 | |
| US7709506B2 | United States of America | B2 | |
| JP2010111699A | Japan | A | |
| JP4472349B2 | Japan | B2 | |
| IL163090A | Israel | A | |
| US2010215652A1 | United States of America | A1 | |
| US2010215661A1 | United States of America | A1 | |
| EP1864975B1 | European Patent Office (EPO) | B1 | |
| AT485275T | Austria | T | |
| DE60334651D1 | Germany | D1 | |
| EP2258687A1 | European Patent Office (EPO) | A1 | |
| PT1864975E | Portugal | E | |
| DK1864975T3 | Denmark | T3 | |
| SI1864975T1 | Slovenia | T1 | |
| ES2352297T3 | Spain | T3 | |
| CA2474192C | Canada | C | |
| KR101058292B1 | Republic of Korea | B1 | |
| US8252818B2 | United States of America | B2 | |
| EP2258687B1 | European Patent Office (EPO) | B1 | |
| PL212910B1 | Poland | B1 | |
| ES2400486T3 | Spain | T3 | |
| US8575204B2 | United States of America | B2 | |
| CY1111083T1 | Cyprus | T1 | |
| BRPI0307351B1 | Brazil | B1 | |
| BRPI0307351B8 | Brazil | B8 |
Numbers
- Publication, DOCDB
- 7337
- Publication, EPODOC
- IS7337
- Application
- 7337
- Application, DOCDB
- 7337
- Application, EPODOC
- IS20040007337
Titles2
- Icelandic
- Nikótínamíð afleiður nytsamlegar sem P38 hindrar
- English
- Nicotinamide derivatives are useful as inhibitors of P38
Classification
- CPC, 55
- C07D213/82
- C07D401/12
- C07D401/14
- C07D405/12
- C07D409/12
- C07D417/12
- A61P1/00
- A61P1/04
- A61P11/00
- A61P11/02
- A61P11/04
- A61P11/06
- A61P11/08
- A61P13/08
- A61P13/12
- A61P15/14
- A61P17/00
- A61P17/02
- A61P17/04
- A61P17/06
- A61P17/08
- A61P19/00
- A61P19/02
- A61P19/04
- A61P19/06
- A61P19/08
- A61P19/10
- A61P21/00
- A61P25/00
- A61P25/04
- A61P25/06
- A61P25/08
- A61P25/14
- A61P25/16
- A61P25/28
- A61P27/02
- A61P27/14
- A61P29/00
- A61P31/00
- A61P31/04
- A61P31/06
- A61P31/08
- A61P31/18
- A61P33/02
- A61P33/06
- A61P35/00
- A61P37/06
- A61P37/08
- A61P39/02
- A61P43/00
- A61P7/02
- A61P9/00
- A61P9/04
- A61P9/10
- A61P3/10
- IPC, 52
- A61K
- A61K31 443
- A61K31 4436
- A61K31 4439
- A61K31 444
- A61K31 496
- A61P
- A61P3 10
- A61P7 02
- A61P9 10
- A61P11 00
- A61P11 02
- A61P11 04
- A61P11 06
- A61P11 08
- A61P13 12
- A61P17 02
- A61P17 04
- A61P17 06
- A61P19 00
- A61P19 02
- A61P19 04
- A61P19 06
- A61P19 08
- A61P19 10
- A61P21 00
- A61P25 00
- A61P25 04
- A61P25 08
- A61P25 14
- A61P25 16
- A61P25 28
- A61P27 14
- A61P29 00
- A61P31 00
- A61P31 04
- A61P31 06
- A61P31 18
- A61P33 02
- A61P33 06
- A61P35 00
- A61P37 06
- A61P37 08
- A61P39 02
- A61P43 00
- C07D
- C07D213 82
- C07D401 12
- C07D401 14
- C07D405 12
- C07D409 12
- C07D417 12