HUT73501A

Microencapsulated 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles

Abstract

Sustained-release microparticle composition. The microparticle composition can be formulated to provide extended release over a period of from about 7 days to about 200 days. The microparticles may be formulated with a biodegradable and biocompatible polymer, and an active agent, such as risperidone, 9-hydroxy-risperidone, and pharmaceutically acceptable acid addition salts of the foregoing.

Term

No projected expiry on record.

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59 members in 31 offices

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Priority claims7

Priority claims
DocumentOfficeKindDate
15440393United States of AmericaA
15440393United States of AmericaA
9403754European Patent Office (EPO)W
9403754European Patent Office (EPO)W
938
US19930154403
WO1994EP03754

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HUT73501AThis recordHungaryA
EP0729357A1European Patent Office (EPO)A1
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CN1137756AChinaA
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CZ293764B6CzechiaB6
US6803055B2United States of AmericaB2
EP0729357B1European Patent Office (EPO)B1
US2005025828A1United States of AmericaA1
ATE288270T1AustriaT1
DE69434258D1GermanyD1
JP3645906B2JapanB2
CL2004001182A1ChileA1
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