HUP0303084A2

17 beta-carbothioate 17-alpha-arylcarbonyloxyloxy androstane derivative as anti-inflammatory agents, process for their preparation and pharmaceutical compositions containing them

Abstract

The subject of the invention is compounds of general formula (I), their salts and solvates - in the formula, R1 is C1-6 alkyl or C1-6 haloalkyl-, R2 is -C(=O)-aryl- or -C(=O)- heteroaryl-, R3 is a hydrogen atom, methyl (this can be in the a or b configuration) or methylene group, R4 and R5 are the same or different and are hydrogen or halogen, and _ _ _ is a single or double bond. The invention also applies to the pharmaceutical preparations containing the compounds of general formula (I) above, to the use of the compounds and pharmaceutical preparations as human and veterinary medicine, to the production process of the compounds, and to the new intermediates used in the production process. HE

HUP0303084A2, drawing sheet 1
Sheet 1 of 15

Term

No projected expiry on record.

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