EP1542996A4
Octahydro-2-h-naphtho 1,2-f indole-4-carboxamide derivatives as selective glucocorticoid receptor modulators
158 sheets
Sheet 1 Sheet 2 Sheet 3 Sheet 4 Sheet 5 Sheet 6 Sheet 7 Sheet 8 Sheet 9 Sheet 10 Sheet 11 Sheet 12 Sheet 13 Sheet 14 Sheet 15 Sheet 16 Sheet 17 Sheet 18 Sheet 19 Sheet 20 Sheet 21 Sheet 22 Sheet 23 Sheet 24 Sheet 25 Sheet 26 Sheet 27 Sheet 28 Sheet 29 Sheet 30 Sheet 31 Sheet 32 Sheet 33 Sheet 34 Sheet 35 Sheet 36 Sheet 37 Sheet 38 Sheet 39 Sheet 40 Sheet 41 Sheet 42 Sheet 43 Sheet 44 Sheet 45 Sheet 46 Sheet 47 Sheet 48 Sheet 49 Sheet 50 Sheet 51 Sheet 52 Sheet 53 Sheet 54 Sheet 55 Sheet 56 Sheet 57 Sheet 58 Sheet 59 Sheet 60 Sheet 61 Sheet 62 Sheet 63 Sheet 64 Sheet 65 Sheet 66 Sheet 67 Sheet 68 Sheet 69 Sheet 70 Sheet 71 Sheet 72 Sheet 73 Sheet 74 Sheet 75 Sheet 76 Sheet 77 Sheet 78 Sheet 79 Sheet 80 Sheet 81 Sheet 82 Sheet 83 Sheet 84 Sheet 85 Sheet 86 Sheet 87 Sheet 88 Sheet 89 Sheet 90 Sheet 91 Sheet 92 Sheet 93 Sheet 94 Sheet 95 Sheet 96 Sheet 97 Sheet 98 Sheet 99 Sheet 100 Sheet 101 Sheet 102 Sheet 103 Sheet 104 Sheet 105 Sheet 106 Sheet 107 Sheet 108 Sheet 109 Sheet 110 Sheet 111 Sheet 112 Sheet 113 Sheet 114 Sheet 115 Sheet 116 Sheet 117 Sheet 118 Sheet 119 Sheet 120 Sheet 121 Sheet 122 Sheet 123 Sheet 124 Sheet 125 Sheet 126 Sheet 127 Sheet 128 Sheet 129 Sheet 130 Sheet 131 Sheet 132 Sheet 133 Sheet 134 Sheet 135 Sheet 136 Sheet 137 Sheet 138 Sheet 139 Sheet 140 Sheet 141 Sheet 142 Sheet 143 Sheet 144 Sheet 145 Sheet 146 Sheet 147 Sheet 148 Sheet 149 Sheet 150 Sheet 151 Sheet 152 Sheet 153 Sheet 154 Sheet 155 Sheet 156 Sheet 157 Sheet 158
Every citation, both ways
| Document | Relation | Office | Category | Cited during | Relevant claims |
|---|---|---|---|---|---|
| EP0102404A1 | Cites | European Patent Office (EPO) | X | Search report | 1-3,5-11,18-21,23-28 |
| EP0102404A | Cites | European Patent Office (EPO) | – | – | – |
| KUMAR V ET AL: "NON-STEROIDAL GLUCOCORTICOID-LIKE SUBSTANCES: RECEPTOR BINDING AND IN VIVO ACTIVITY", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US, vol. 36, 1 January 1993 (1993-01-01), pages 3278 - 3285, XP001019064, ISSN: 0022-2623 | Non-patent | – | – | Search report | – |
| PHILIP SCHANE H ET AL: "Glucocorticoid/Antiinflammatory activities of nonsteroidal phenylpyrazoles in the rat", STEROIDS, ELSEVIER SCIENCE PUBLISHERS, NEW YORK, NY, US, vol. 45, no. 2, 1 February 1985 (1985-02-01), pages 171 - 185, XP023431680, ISSN: 0039-128X, [retrieved on 19850201] | Non-patent | – | – | Search report | – |
11 members in 6 offices
Priority claims5
| Document | Office | Kind | Date |
|---|---|---|---|
| 412231P | United States of America | – | |
| 41223102 | United States of America | P | |
| 476079P | United States of America | – | |
| 47607903 | United States of America | P | |
| 0329494 | United States of America | W |
Members11
| Document | Office | Kind | |
|---|---|---|---|
| CA2499150A1 | Canada | A1 | |
| WO2004026248A2 | World Intellectual Property Organization (WIPO) | A2 | |
| AU2003270783A1 | Australia | A1 | |
| WO2004026248A3 | World Intellectual Property Organization (WIPO) | A3 | |
| EP1542996A2 | European Patent Office (EPO) | A2 | |
| US2005245588A1 | United States of America | A1 | |
| JP2006503107A | Japan | A | |
| EP1542996A4This record | European Patent Office (EPO) | A4 | |
| AU2003270783B2 | Australia | B2 | |
| AU2003270783C1 | Australia | C1 | |
| JP4520309B2 | Japan | B2 |
16 legal events, as the office reported them to INPADOC
Over the term
Point at a mark for the eventEvents
| Event | Code | |
|---|---|---|
| Application deemed to be withdrawnWithdrawn18D | 18D | |
| Information on the status of an ep patent application or granted ep patentGrantedSTATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWNSTAA | STAA | |
| First examination report despatched17Q | 17Q | |
| Party data changed (applicant data changed or rights of an application transferred)RAP1 | RAP1 | |
| Supplementary search report drawn up and despatchedA4 | A4 | |
| Information provided on ipc code assigned before grantRIC1 | RIC1 | |
| Information provided on ipc code assigned before grantRIC1 | RIC1 | |
| Information provided on ipc code assigned before grantRIC1 | RIC1 | |
| Information provided on ipc code assigned before grantRIC1 | RIC1 | |
| Information provided on ipc code assigned before grantRIC1 | RIC1 | |
| Requested extension states of the european patent have changedRAX | RAX | |
| Requested extension states of the european patent have changedRAX | RAX | |
| Request for examination filed17P | 17P | |
| Designated contracting statesAK | AK | |
| Request for extension of the european patentAX | AX | |
| Public reference made under article 153(3) epc to a published international application that has entered the european phaseORIGINAL CODE: 0009012PUAI | PUAI |
Numbers
- Publication
- 1542996
- Application
- 37524956
Titles3
- German
- OCTAHYDRO-2H-NAPHTOç1,2-F INDOL-4-CARBONSûUREAMIDDERIVATE ALS SELEKTIVE MODULATOREN DES GLUCOCORTICOIDREZEPTORS
- English
- OCTAHYDRO-2-H-NAPHTHO 1,2-F INDOLE-4-CARBOXAMIDE DERIVATIVES AS SELECTIVE GLUCOCORTICOID RECEPTOR MODULATORS
- French
- DERIVES D'OCTAHYDRO-2-H-NAPHTHO 1,2-F INDOLE-4-CARBOXAMIDE EN TANT QUE MODULATEURS SELECTIFS DE RECEPTEUR GLUCOCORTICOIDE
Classification
- CPC, 54
- C07J71/0047
- C07D231/54
- C07D401/12
- C07D403/04
- C07D409/12
- C07D413/04
- C07D417/04
- C07D491/113
- A61P1/04
- A61P1/16
- A61P11/00
- A61P11/02
- A61P11/06
- A61P17/00
- A61P17/02
- A61P17/04
- A61P17/06
- A61P17/10
- A61P17/14
- A61P19/00
- A61P19/02
- A61P21/00
- A61P25/00
- A61P25/18
- A61P25/20
- A61P25/22
- A61P25/24
- A61P25/28
- A61P27/02
- A61P29/00
- A61P3/02
- A61P3/04
- A61P3/14
- A61P31/08
- A61P31/18
- A61P35/00
- A61P35/02
- A61P3/06
- A61P37/02
- A61P37/04
- A61P37/06
- A61P37/08
- A61P39/02
- A61P43/00
- A61P5/28
- A61P5/38
- A61P5/40
- A61P5/42
- A61P5/46
- A61P7/00
- A61P7/04
- A61P7/10
- A61P9/00
- A61P9/14
- IPC, 9
- C07J71 00
- A61K
- A61K31 415
- A61K31 4162
- A61K31 58
- A61P5 46
- C07D231 44
- C07D231 54
- C07D417 00
Designated states29
- Contracting states, 27
- Austria
- Belgium
- Bulgaria
- Switzerland
- Cyprus
- Czechia
- Germany
- Denmark
- Estonia
- Spain
- Finland
- France
- United Kingdom
- Greece
- Hungary
- Ireland
- Italy
- Liechtenstein
- Luxembourg
- Monaco
- Netherlands (Kingdom of the)
- Portugal
- Romania
- Sweden
and 3 moreShow fewer
- Slovenia
- Slovakia
- Türkiye
- Extension states, 2
- Lithuania
- Latvia
