EP0404283A3
11-beta-aryl-4-estrene, method for its production and its use as a medicine
Abstract
Compounds of general formula I have been described wherein X, R¹, R², R³ and R⁴ have the meaning given in the description, as well as processes for their preparation, pharmaceutical compositions containing them and their use for the treatment of diseases. Above all, the compounds possess antigestagenic and antiglucocorticoid activity.

Term
Term ended
Projected expiry passed 1 June 2010, 16.3 years ago.
- Priority
- Filed
- Published
- Projected expiry
- Today
1 sheet
Sheet 1
Every citation, both ways
| Document | Relation | Office | Category | Cited during |
|---|---|---|---|---|
| EP0192598A2 | Cites | European Patent Office (EPO) | A | Search report |
| EP0196707A1 | Cites | European Patent Office (EPO) | X | Search report |
| EP0277089A1 | Cites | European Patent Office (EPO) | Y | Search report |
| EP0308345A1 | Cites | European Patent Office (EPO) | Y | Search report |
| AU59584A | Cites | Australia | A | Search report |
| WO8705908A1 | Cites | World Intellectual Property Organization (WIPO) | Y | Search report |
| WO8801868A1 | Cites | World Intellectual Property Organization (WIPO) | A | Search report |
39 members in 19 offices
Priority claims4
| Document | Office | Kind | Date |
|---|---|---|---|
| 3921059 | Germany | A | |
| 3921059 | Germany | A | |
| 3921059 | Germany | – | |
| DE19893921059 | – | – | – |
Members39
| Document | Office | Kind | |
|---|---|---|---|
| NO902800D0 | Norway | D0 | |
| HU903961D0 | Hungary | D0 | |
| CA2019404A1 | Canada | A1 | |
| IE902280L | Ireland | L | |
| EP0404283A2 | European Patent Office (EPO) | A2 | |
| NO902800L | Norway | L | |
| CN1048219A | China | A | |
| AU5778090A | Australia | A | |
| DE3921059A1 | Germany | A1 | |
| IE902280A1 | Ireland | A1 | |
| PT94462A | Portugal | A | |
| HUT54705A | Hungary | A | |
| IL94819D0 | Israel | D0 | |
| ZA904893B | South Africa | B | |
| JPH03128323A | Japan | A | |
| EP0404283A3This record | European Patent Office (EPO) | A3 | |
| DD295639A5 | German Democratic Republic (until 1990) | A5 | |
| AU640664B2 | Australia | B2 | |
| HU209949B | Hungary | B | |
| IL94819A | Israel | A | |
| FI954748A | Finland | A | |
| NO178768B | Norway | B | |
| EP0404283B1 | European Patent Office (EPO) | B1 | |
| AT137762T | Austria | T | |
| NO178768C | Norway | C | |
| DE59010312D1 | Germany | D1 | |
| GR3020098T3 | Greece | T3 | |
| DK0404283T3 | Denmark | T3 | |
| ES2088959T3 | Spain | T3 | |
| CN1133296A | China | A | |
| IE74191B1 | Ireland | B1 | |
| US5728689A | United States of America | A | |
| US5843933A | United States of America | A | |
| JP2911553B2 | Japan | B2 | |
| CN1048499C | China | C | |
| CN1061052C | China | C | |
| FI110688B | Finland | B | |
| CA2019404C | Canada | C | |
| FI111844B | Finland | B |
58 legal events, as 7 offices reported them to INPADOC
Over the term
Point at a mark for the eventEvents
| Event | Code | Office | |
|---|---|---|---|
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Announcement of lapse in spainLapsedFD2A | FD2A | ES | |
| Notification of lapseLapsedST | ST | FR | |
| Nl: lapsed or anulled due to non-payment of the annual feeLapsedNLV4 | NLV4 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Patent ceasedCeasedPL | PL | CH | |
| Ep patent lapsedLapsedEBP | EBP | DK | |
| Se: european patent has lapsedLapsedEUG | EUG | EP | |
| Gb: european patent ceased through non-payment of renewal feeCeasedGBPC | GBPC | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Be: lapsedLapsedBERE | BERE | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| European patent in force as of 2002-01-01IF02 | IF02 | GB | |
| No opposition filedOpposition26N | 26N | EP | |
| No opposition filed within time limitOppositionORIGINAL CODE: 0009261PLBE | PLBE | EP | |
| Information on the status of an ep patent application or granted ep patentGrantedSTATUS: NO OPPOSITION FILED WITHIN TIME LIMITSTAA | STAA | EP | |
| Definitive protectionFG2A | FG2A | ES | |
| Definitive protectionFG2A | FG2A | ES | |
| Fr: translation filedET | ET | EP | |
| Ep patent with danish claimsT3 | T3 | DK | |
| Gb: translation of ep patent filed (gb section 77(6)(a)/1977)GBT | GBT | EP | |
| Validation in greece3020098FG4A | FG4A | GR | |
| It: translation for a ep patent filedITF | ITF | EP | |
| It: translation for a ep patent filedITF | ITF | EP | |
| New agentNV | NV | CH | |
| Corresponds to:REF | REF | EP | |
| Designated contracting statesAK | AK | EP | |
| Corresponds to:REF | REF | EP | |
| (expected) grantORIGINAL CODE: 0009210GRAA | GRAA | EP | |
| Despatch of communication of intention to grant a patentORIGINAL CODE: EPIDOS IGRAGRAH | GRAH | EP | |
| First examination report despatched17Q | 17Q | EP | |
| Designated contracting statesAK | AK | EP | |
| Search report despatchedORIGINAL CODE: 0009013PUAL | PUAL | EP | |
| Request for examination filed17P | 17P | EP | |
| Designated contracting statesAK | AK | EP | |
| Public reference made under article 153(3) epc to a published international application that has entered the european phaseORIGINAL CODE: 0009012PUAI | PUAI | EP |
Numbers
- Publication
- 0404283
- Publication, DOCDB
- 0404283
- Publication, EPODOC
- EP0404283
- Application
- 250142
- Application, DOCDB
- 90250142
- Application, EPODOC
- EP19900250142
Titles3
- German
- 11-Beta-aryl-4-estrene, Verfahren zu ihrer Herstellung sowie deren Verwendung als Arzneimittel
- English
- 11-Beta-aryl-4-estrene, method for its production and its use as a medicine
- French
- 11-Bêta-aryl-4-estrène, son procédé de préparation et son application comme médicament
Classification
- CPC, 14
- C07J1/0096
- C07J1/0085
- C07J1/0092
- C07J17/00
- C07J41/0083
- C07J41/0094
- C07J43/003
- A61P13/02
- A61P15/00
- A61P27/02
- A61P3/00
- A61P5/36
- A61P9/10
- A61P9/12
- IPC, 18
- A61K31 565
- A61K31 56
- A61P3 00
- A61P9 10
- A61P9 12
- A61P13 02
- A61P15 00
- A61P27 02
- C07J1 00
- C07J3 00
- C07J5 00
- C07J7 00
- C07J9 00
- C07J17 00
- C07J19 00
- C07J21 00
- C07J41 00
- C07J43 00
Designated states1
- Contracting states, 1
- Sweden