Pharmaceutical formulations of acid labile substances for oral use
Abstract
Pharmaceutical preparation containing an acid labile compound together with an alkaline reacting compound or an alkaline salt of an acid labile compound optionally together with an alkaline compound as the core material, one or more subcoating layers comprising inert reacting compounds which are soluble or rapidly disintegrating in water, or polymeric, water soluble filmforming compounds, optionally containing pH-buffering alkaline compounds and an enteric coating as well as a process for the preparation thereof and the use in the treatment of gastrointestinal diseases.
Term
Term ended
Projected expiry passed 16 April 2007, 19.4 years ago.
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Every citation, both waysCites: the store holds 7 of 8
| Document | Relation | Office | Category | Cited during |
|---|---|---|---|---|
| EP0080602A1 | Cites | European Patent Office (EPO) | YD | Search report |
| EP0124495A2 | Cites | European Patent Office (EPO) | X | Search report |
| EP0173664A2 | Cites | European Patent Office (EPO) | XD | Search report |
| GB1190387A | Cites | United Kingdom | A | Search report |
| FR2272639A1 | Cites | France | Y | Search report |
| DE3233764A1 | Cites | Germany | A | Search report |
| GB760403A | Cites | United Kingdom | Y | Search report |
| PATENT ABSTRACTS OF JAPAN, vol. 8, no. 106 (C-223)[1543], 18th May 1984; & JP-A-59 020 219 (SHINETSU KAGAKU KOGYO K.K.) 01-02-1984 | Non-patent | – | – | Search report |
82 members in 37 offices
Priority claims5
| Document | Office | Kind | Date |
|---|---|---|---|
| 8610573 | United Kingdom | A | |
| 8610573 | United Kingdom | A | |
| 8610573 | United Kingdom | – | |
| 8610573 | – | – | – |
| GB19860010573 | – | – | – |
Members82
| Document | Office | Kind | |
|---|---|---|---|
| GB8610573D0 | United Kingdom | D0 | |
| CY1860A | Cyprus | A | |
| DK215987D0 | Denmark | D0 | |
| NO871791D0 | Norway | D0 | |
| PT84786A | Portugal | A | |
| IE871106L | Ireland | L | |
| DK215987A | Denmark | A | |
| FI871914A | Finland | A | |
| IS3222A7 | Iceland | A7 | |
| NO871791L | Norway | L | |
| EP0244380A2 | European Patent Office (EPO) | A2 | |
| GB2189699A | United Kingdom | A | |
| AU7192287A | Australia | A | |
| JPS62258316A | Japan | A | |
| CN87103285A | China | A | |
| KR870009718A | Republic of Korea | A | |
| ZA872379B | South Africa | B | |
| HUT44171A | Hungary | A | |
| PL265417A1 | Poland | A1 | |
| YU68087A | Yugoslavia, later Serbia and Montenegro (until 2006) | A | |
| EP0244380A3This record | European Patent Office (EPO) | A3 | |
| CS307387A2 | Czechoslovakia (until 1993) | A2 | |
| US4853230A | United States of America | A | |
| HU198385B | Hungary | B | |
| ES2010648A4 | Spain | A4 | |
| PT84786B | Portugal | B | |
| DE244380T1 | Germany | T1 | |
| CS268535B2 | Czechoslovakia (until 1993) | B2 | |
| GR890300156T1 | Greece | T1 | |
| NZ220097A | New Zealand | A | |
| PH24440A | Philippines | A | |
| AU603568B2 | Australia | B2 | |
| SU1709894A3 | Soviet Union (until 1991) | A3 | |
| CA1302891C | Canada | C | |
| EP0502556A1 | European Patent Office (EPO) | A1 | |
| MY102675A | Malaysia | A | |
| EP0244380B1 | European Patent Office (EPO) | B1 | |
| AT84211T | Austria | T | |
| ATE84211T1 | Austria | T1 | |
| DE3783386D1 | Germany | D1 | |
| EG18517A | Egypt | A | |
| DE3783386T2 | Germany | T2 | |
| GR3007448T3 | Greece | T3 | |
| AR243377A1 | Argentina | A1 | |
| EP0565210A2 | European Patent Office (EPO) | A2 | |
| YU46421B | Yugoslavia, later Serbia and Montenegro (until 2006) | B | |
| LT2260B | Lithuania | B | |
| LV5393A3 | Latvia | A3 | |
| FI91708B | Finland | B | |
| NO174952B | Norway | B | |
| CN1025151C | China | C | |
| ES2010648T3 | Spain | T3 | |
| FI91708C | Finland | C | |
| NO174952C | Norway | C | |
| JPH0667837B2 | Japan | B2 | |
| IE61837B1 | Ireland | B1 | |
| DK169987B1 | Denmark | B1 | |
| KR950004886B1 | Republic of Korea | B1 | |
| EP0565210A3 | European Patent Office (EPO) | A3 | |
| HRP920855A2 | Croatia | A2 | |
| HK104095A | Hong Kong, China | A | |
| EP0502556B1 | European Patent Office (EPO) | B1 | |
| AT139692T | Austria | T | |
| ATE139692T1 | Austria | T1 | |
| DE3751851D1 | Germany | D1 | |
| ES2089277T3 | Spain | T3 | |
| DE3751851T2 | Germany | T2 | |
| GR3020501T3 | Greece | T3 | |
| LV5753A4 | Latvia | A4 | |
| SI8710680A | Slovenia | A | |
| HK55497A | Hong Kong, China | A | |
| LV5753B4 | Latvia | B4 | |
| SI8710680B | Slovenia | B | |
| DD260222B5 | German Democratic Republic (until 1990) | B5 | |
| HRP920855B1 | Croatia | B1 | |
| EP0565210B1 | European Patent Office (EPO) | B1 | |
| AT186639T | Austria | T | |
| ATE186639T1 | Austria | T1 | |
| ES2137966T3 | Spain | T3 | |
| GR3032639T3 | Greece | T3 | |
| IS1918B | Iceland | B | |
| DZ1078A1 | Algeria | A1 |
110 legal events, as 5 offices reported them to INPADOC
Over the term
Point at a mark for the eventEvents
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|---|---|---|---|
| Opposition filed (corrected)OppositionR26 | R26 | EP | |
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| Opposition data, opponent's data or that of the opponent's representative modifiedOppositionORIGINAL CODE: 0009299OPPOPLAB | PLAB | EP | |
| Be: patent expiredExpiredBE20 | BE20 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Announcement of lapse in spainLapsedFD2A | FD2A | ES | |
| Se: european patent has lapsedLapsedEUG | EUG | EP | |
| Nl: ceased due to reaching the maximum lifetime of a patentCeasedNLV7 | NLV7 | EP | |
| Patent ceasedCeasedPL | PL | CH | |
| Patent expired after termination of 20 yearsExpiredPE20 | PE20 | GB | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Lapsed in a contracting state [announced via postgrant information from national office to epo]LapsedPG25 | PG25 | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
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| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| Annual fee paid to national office [announced via postgrant information from national office to epo]GrantedPGFP | PGFP | EP | |
| European patent in force as of 2002-01-01IF02 | IF02 | GB | |
| Nl: decision of oppositionOppositionNLR2 | NLR2 | EP | |
| Opposition proceedings terminatedOpposition27C | 27C | EP | |
| Termination of opposition procedure: date of legal effect publishedOppositionORIGINAL CODE: 0009276PLBM | PLBM | EP | |
| Information on the status of an ep patent application or granted ep patentGrantedSTATUS: OPPOSITION PROCEDURE CLOSEDSTAA | STAA | EP | |
| Opposition procedure terminatedOppositionORIGINAL CODE: EPIDOS OPPCPLBL | PLBL | EP | |
| Amendments to the register in respect of changes of name or changes affecting rights (sect. 32/1977)732E | 732E | GB | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
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| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
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| Opposition filedOppositionORIGINAL CODE: 0009260PLBI | PLBI | EP | |
| Se: european patent in force in swedenEAL | EAL | EP | |
| Lu: last paid annual feeEPTA | EPTA | EP | |
| Definitive protectionFG2A | FG2A | ES | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
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| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
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| Opposition filedOppositionORIGINAL CODE: 0009260PLBI | PLBI | EP | |
| Opposition filedOppositionORIGINAL CODE: 0009260PLBI | PLBI | EP | |
| Opposition filedOppositionORIGINAL CODE: 0009260PLBI | PLBI | EP | |
| Amendments to the register in respect of changes of name or changes affecting rights (sect. 32/1977)732E | 732E | GB | |
| Validation in greece3007448FG4A | FG4A | GR | |
| Nl: opposition has been filed with the epoOppositionNLR1 | NLR1 | EP | |
| Opposition filed (corrected)OppositionR26 | R26 | EP | |
| Opposition filedOpposition26 | 26 | EP | |
| Fr: translation filedET | ET | EP | |
| Corresponds to:REF | REF | EP | |
| It: translation for a ep patent filedITF | ITF | EP | |
| It: translation for a ep patent filedITF | ITF | EP | |
| Opposition data, opponent's data or that of the opponent's representative modifiedOppositionORIGINAL CODE: 0009299OPPOPLAB | PLAB | EP | |
| Opposition filedOppositionORIGINAL CODE: 0009260PLBI | PLBI | EP | |
| Licence recorded0100 LABORATOIRES ASTRA FRANCE111L | 111L | EP | |
| Designated contracting statesAK | AK | EP | |
| Corresponds to:REF | REF | EP | |
| Miscellaneous (additional remarks)TEILANMELDUNG 92107178.3 EINGEREICHT AM 16/04/87.XX | XX | EP | |
| (expected) grantORIGINAL CODE: 0009210GRAA | GRAA | EP | |
| Fr: translation or corrected translation of claims filedEL1 | EL1 | EP | |
| First examination report despatched17Q | 17Q | EP |
Numbers
- Publication
- 0244380
- Publication, DOCDB
- 0244380
- Publication, EPODOC
- EP0244380
- Application
- 87850126
- Application, DOCDB
- 87850126
- Application, EPODOC
- EP19870850126
Titles3
- English
- Pharmaceutical formulations of acid labile substances for oral use
- French
- Formulations pharmaceutiques de substances sensibles aux acides pour utilisation orale
- German
- Arzneiformulierungen säurelabiler Substanzen zur oralen Verwendung
Classification
- CPC, 5
- A61K31/415
- A61K9/2009
- A61K9/2886
- A61K9/5073
- A61K31/44
- IPC, 11
- A61K31 415
- A61K9 16
- A61K9 20
- A61K9 28
- A61K9 30
- A61K9 32
- A61K9 50
- A61K9 52
- A61K9 54
- A61K31 433
- A61K31 44
Designated states1
- Contracting states, 1
- Sweden