ECSP12012218A
Piperidin-4-yl azetidine derivatives as jak1 inhibitors
Abstract
The present invention provides piperidin-4-yl azetidine derivatives, as well as its compositions and methods of use, which modulate the activity of Janus kinase (JAK1) and are useful in the treatment of diseases related to the activity of JAK1 which includes, by For example, inflammatory disorders, autoimmune disorders, cancer, and other diseases.
Term
No projected expiry on record.
- Priority
- Filed
- Published
- Today
141 members in 39 offices
Priority claims2
| Document | Office | Kind | Date |
|---|---|---|---|
| 31258810 | United States of America | P | |
| 41560210 | United States of America | P |
Members141
| Document | Office | Kind | |
|---|---|---|---|
| CA2792508A1 | Canada | A1 | |
| US2011224190A1 | United States of America | A1 | |
| WO2011112662A1 | World Intellectual Property Organization (WIPO) | A1 | |
| TW201206923A | Taiwan Province of China | A | |
| AR081315A1 | Argentina | A1 | |
| AU2011224484A1 | Australia | A1 | |
| SG183551A1 | Singapore | A1 | |
| PH12012501768A1 | Philippines | A1 | |
| MX2012010344A | Mexico | A | |
| ECSP12012218AThis record | Ecuador | A | |
| CL2012002501A1 | Chile | A1 | |
| CR20120510A | Costa Rica | A | |
| EP2545045A1 | European Patent Office (EPO) | A1 | |
| CO6602158A2 | Colombia | A2 | |
| PE20130038A1 | Peru | A1 | |
| CN102985417A | China | A | |
| KR20130038834A | Republic of Korea | A | |
| EA201290894A1 | Eurasian Patent Organization (EAPO) | A1 | |
| JP2013522214A | Japan | A | |
| HK1177741A | Hong Kong, China | A | |
| HK1177741A1 | Hong Kong, China | A1 | |
| ZA201207420B | South Africa | B | |
| US8765734B2 | United States of America | B2 | |
| NZ602313A | New Zealand | A | |
| US2014275031A1 | United States of America | A1 | |
| CN102985417B | China | B | |
| AU2015205858A1 | Australia | A1 | |
| UA110108C2 | Ukraine | C2 | |
| EP2545045B1 | European Patent Office (EPO) | B1 | |
| DK2545045T3 | Denmark | T3 | |
| MX336932B | Mexico | B | |
| JP5858484B2 | Japan | B2 | |
| TWI531572B | Taiwan Province of China | B | |
| ES2569539T3 | Spain | T3 | |
| HRP20160326T1 | Croatia | T1 | |
| JP2016094443A | Japan | A | |
| SI2545045T1 | Slovenia | T1 | |
| SMT201600085B | San Marino | B | |
| EP3050882A1 | European Patent Office (EPO) | A1 | |
| BR112012022513A2 | Brazil | A2 | |
| PL2545045T3 | Poland | T3 | |
| ME02386B | Montenegro | B | |
| US9464088B2 | United States of America | B2 | |
| IL221823A | Israel | A | |
| RS54823B1 | Serbia | B1 | |
| TW201638088A | Taiwan Province of China | A | |
| HUE028723T2 | Hungary | T2 | |
| AU2017201801A1 | Australia | A1 | |
| AU2015205858B2 | Australia | B2 | |
| PH12015502575A1 | Philippines | A1 | |
| PH12015502575B1 | Philippines | B1 | |
| CY1117435T1 | Cyprus | T1 | |
| MX347851B | Mexico | B | |
| JP6158282B2 | Japan | B2 | |
| TWI592413B | Taiwan Province of China | B | |
| JP2017149779A | Japan | A | |
| US2017246157A1 | United States of America | A1 | |
| TW201734014A | Taiwan Province of China | A | |
| CA2792508C | Canada | C | |
| EP3050882B1 | European Patent Office (EPO) | B1 | |
| MX354212B | Mexico | B | |
| DK3050882T3 | Denmark | T3 | |
| ES2662588T3 | Spain | T3 | |
| PT3050882T | Portugal | T | |
| JP6318291B2 | Japan | B2 | |
| KR101857680B1 | Republic of Korea | B1 | |
| KR20180054890A | Republic of Korea | A | |
| LT3050882T | Lithuania | T | |
| HRP20180552T1 | Croatia | T1 | |
| US9999619B2 | United States of America | B2 | |
| SI3050882T1 | Slovenia | T1 | |
| NO3050882T3 | Norway | T3 | |
| SMT201800137T1 | San Marino | T1 | |
| EA030376B1 | Eurasian Patent Organization (EAPO) | B1 | |
| RS57219B1 | Serbia | B1 | |
| EP3354652A1 | European Patent Office (EPO) | A1 | |
| JP2018118992A | Japan | A | |
| HUE037077T2 | Hungary | T2 | |
| PL3050882T3 | Poland | T3 | |
| ME03002B | Montenegro | B | |
| KR101911697B1 | Republic of Korea | B1 | |
| KR20180117206A | Republic of Korea | A | |
| TWI643857B | Taiwan Province of China | B | |
| CY1120154T1 | Cyprus | T1 | |
| US2018353499A1 | United States of America | A1 | |
| TW201906613A | Taiwan Province of China | A | |
| MX364636B | Mexico | B | |
| MX2019005232A | Mexico | A | |
| AU2017201801B2 | Australia | B2 | |
| EA201890558A1 | Eurasian Patent Organization (EAPO) | A1 | |
| AU2019257385A1 | Australia | A1 | |
| HK1258929A | Hong Kong, China | A | |
| HK1258929A1 | Hong Kong, China | A1 | |
| KR20200033996A | Republic of Korea | A | |
| EP3354652B1 | European Patent Office (EPO) | B1 | |
| DK3354652T3 | Denmark | T3 | |
| TWI694826B | Taiwan Province of China | B | |
| MY175156A | Malaysia | A | |
| US10695337B2 | United States of America | B2 | |
| PT3354652T | Portugal | T |
Showing 100 of 141
Numbers
- Publication
- 2012012218
- Application
- 1218
Titles2
- English
- DERIVATIVES OF PIPERIDIN-4-IL AZETIDINE AS INHIBITORS OF JAK1
- Spanish
- DERIVADOS DE PIPERIDIN-4-IL AZETIDINA COMO INHIBIDORES DE JAK1
Classification
- CPC, 23
- A61K31/4545
- C07D487/04
- A61K31/519
- A61P27/02
- A61P11/00
- A61P11/06
- A61P35/00
- A61P19/08
- A61P37/00
- A61P29/00
- A61P19/02
- C07D471/04
- C07D519/00
- C07B2200/13
- A61P1/00
- A61P17/04
- A61P37/06
- C07D401/14
- C07D405/14
- A61K9/0014
- A61K9/0019
- A61K9/0024
- A61K9/0048
- IPC, 6
- C07D401 14
- A61K31 4155
- A61K31 437
- A61K31 4468
- A61P29 00
- C07D405 14