AT307123T
Synthesis of epothilones, intermediates thereto and analogues therof
Abstract
(57) Summary book invention offers the convergence method for preparing EPO チロン A and B which can be used for the medical treatment of Gang who produced Gang and a drug-resistant phenotype, デオキシエポチロン, B, and its analog. Moreover, the intermediate field which can be used in order to prepare the above-mentioned EPO チロン are also offered.
Term
No projected expiry on record.
- Priority
- Filed
- Granted
- Today
77 members in 13 offices
Priority claims4
| Document | Office | Kind | Date |
|---|---|---|---|
| 7594798 | United States of America | P | |
| 9231998 | United States of America | P | |
| 9773398 | United States of America | P | |
| 9904008 | United States of America | W |
Members77
| Document | Office | Kind | |
|---|---|---|---|
| CA2273083A1 | Canada | A1 | |
| WO9901124A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU5792998A | Australia | A | |
| ZA9711282B | South Africa | B | |
| WO9901124A9 | World Intellectual Property Organization (WIPO) | A9 | |
| ZA991497B | South Africa | B | |
| CA2322157A1 | Canada | A1 | |
| WO9943653A1 | World Intellectual Property Organization (WIPO) | A1 | |
| AU2785899A | Australia | A | |
| EP0977563A1 | European Patent Office (EPO) | A1 | |
| EP1058679A1 | European Patent Office (EPO) | A1 | |
| US6204388B1 | United States of America | B1 | |
| EP0977563A4 | European Patent Office (EPO) | A4 | |
| US6242469B1 | United States of America | B1 | |
| JP2001507716A | Japan | A | |
| US6284781B1 | United States of America | B1 | |
| CA2401800A1 | Canada | A1 | |
| WO0164650A2 | World Intellectual Property Organization (WIPO) | A2 | |
| AU4337201A | Australia | A | |
| US6300355B1 | United States of America | B1 | |
| IL138113D0 | Israel | D0 | |
| US6316630B1 | United States of America | B1 | |
| US2002002194A1 | United States of America | A1 | |
| JP2002504540A | Japan | A | |
| US6369234B1 | United States of America | B1 | |
| WO0164650A3 | World Intellectual Property Organization (WIPO) | A3 | |
| US2002058286A1 | United States of America | A1 | |
| US2002058817A1 | United States of America | A1 | |
| EP1058679A4 | European Patent Office (EPO) | A4 | |
| TW504511B | Taiwan Province of China | B | |
| MXPA00008365A | Mexico | A | |
| EP1259490A2 | European Patent Office (EPO) | A2 | |
| AU756699B2 | Australia | B2 | |
| AU758526B2 | Australia | B2 | |
| US2003069277A1 | United States of America | A1 | |
| US2003105330A1 | United States of America | A1 | |
| US2003125362A1 | United States of America | A1 | |
| US6603023B2 | United States of America | B2 | |
| US2003171596A1 | United States of America | A1 | |
| NZ506742A | New Zealand | A | |
| US2003208080A1 | United States of America | A1 | |
| US6656961B2 | United States of America | B2 | |
| JP2004500388A | Japan | A | |
| US2004019089A1 | United States of America | A1 | |
| EP1386922A2 | European Patent Office (EPO) | A2 | |
| US2004044221A1 | United States of America | A1 | |
| EP1386922A3 | European Patent Office (EPO) | A3 | |
| US6723854B2 | United States of America | B2 | |
| US2004102495A1 | United States of America | A1 | |
| US6828340B2 | United States of America | B2 | |
| US2004260098A1 | United States of America | A1 | |
| US6849651B2 | United States of America | B2 | |
| US2005033059A1 | United States of America | A1 | |
| US2005043376A1 | United States of America | A1 | |
| US6867305B2 | United States of America | B2 | |
| EP0977563B1 | European Patent Office (EPO) | B1 | |
| EP1058679B1 | European Patent Office (EPO) | B1 | |
| AT307123TThis record | Austria | T | |
| ATE307123T1 | Austria | T1 | |
| US6965034B2 | United States of America | B2 | |
| US6972335B2 | United States of America | B2 | |
| DE69734362D1 | Germany | D1 | |
| DE69927790D1 | Germany | D1 | |
| DE69734362T2 | Germany | T2 | |
| DE69927790T2 | Germany | T2 | |
| IL138113A | Israel | A | |
| US2008004450A1 | United States of America | A1 | |
| JP2009298816A | Japan | A | |
| US7750164B2 | United States of America | B2 | |
| US2010240721A1 | United States of America | A1 | |
| JP4579351B2 | Japan | B2 | |
| USRE41990E | United States of America | E | |
| US2011263663A1 | United States of America | A1 | |
| EP1386922B1 | European Patent Office (EPO) | B1 | |
| CA2322157C | Canada | C | |
| CA2273083C | Canada | C | |
| US8481575B2 | United States of America | B2 |
1 legal event, as the office reported them to INPADOC
Events
| Event | Code | |
|---|---|---|
| Ceased as to paragraph 5 lit. 3 law introducing patent treatiesCeasedRER | RER |
Numbers
- Application
- 99908420
Titles2
- German
- SYNTHESE VON EPOTHILONEN, IHREN ZWISCHENPRODUKTEN UND ANALOGEN VERBINDUNGEN
- English
- SYNTHESIS OF EPOTHILONES, ITS INTERMEDIATE PRODUCTS AND ANALOGICAL COMPOUNDS
Classification
- CPC, 8
- C07D417/06
- A61P35/00
- C07C59/76
- C07C69/738
- C07D277/24
- C07D313/00
- C07D493/04
- C07F7/1892
- IPC, 16
- A61K31 365
- A61K31 427
- A61P35 00
- C07C59 185
- C07C59 76
- C07C69 66
- C07C69 738
- C07D233 54
- C07D277 24
- C07D277 28
- C07D277 30
- C07D313 00
- C07D417 06
- C07D493 04
- C07F7 02
- C07F7 18