AP3339A
Benzodioxane inhibitors of leukotriene production
Abstract
The present invention relates to compounds of formula (I), wherein R1 to R3, A, X and n are as defined herein. Compounds are useful as leukotriene A4 hydrolase (LTA4H) inhibitors of Formula (I) and for the treatment of disorders associated with LTA4H. The present invention also relates to a compound comprising formula (I) in pharmaceutical compositions, the use of these compounds in the treatment of various diseases and disorders, and a method for preparing these compounds.

Term
No projected expiry on record.
- Priority
- Filed
- Granted
- Today
2 sheets
Sheet 1 Sheet 2
Every citation, both waysCites: the store holds 1 of 2
| Document | Relation | Office | Cited during |
|---|---|---|---|
| US4918092A | Cites | United States of America | Search report |
43 members in 26 offices
Priority claims2
| Document | Office | Kind | Date |
|---|---|---|---|
| 201161452329 | United States of America | P | |
| 2012028843 | United States of America | W |
Members43
| Document | Office | Kind | |
|---|---|---|---|
| CA2835617A1 | Canada | A1 | |
| WO2012125598A1 | World Intellectual Property Organization (WIPO) | A1 | |
| UY33950A | Uruguay | A | |
| TW201302723A | Taiwan Province of China | A | |
| US2013196973A1 | United States of America | A1 | |
| AU2012229172A1 | Australia | A1 | |
| AP2013007044A0 | African Regional Intellectual Property Organization (ARIPO) | A0 | |
| IL227805A0 | Israel | A0 | |
| US8551982B2 | United States of America | B2 | |
| CO6771439A2 | Colombia | A2 | |
| MX2013010457A | Mexico | A | |
| SG193454A1 | Singapore | A1 | |
| CN103415513A | China | A | |
| US2013345195A1 | United States of America | A1 | |
| EP2686310A1 | European Patent Office (EPO) | A1 | |
| KR20140021600A | Republic of Korea | A | |
| EA201301019A1 | Eurasian Patent Organization (EAPO) | A1 | |
| MA35089B1 | Morocco | B1 | |
| JP2014511826A | Japan | A | |
| JP5640162B2 | Japan | B2 | |
| TN2013000362A1 | Tunisia | A1 | |
| NZ614109A | New Zealand | A | |
| AP3339AThis record | African Regional Intellectual Property Organization (ARIPO) | A | |
| GEP20156347B | Georgia | B | |
| US9133146B2 | United States of America | B2 | |
| CN103415513B | China | B | |
| EA023876B1 | Eurasian Patent Organization (EAPO) | B1 | |
| TWI551593B | Taiwan Province of China | B | |
| BR112013023517A2 | Brazil | A2 | |
| AU2012229172B2 | Australia | B2 | |
| IL227805A | Israel | A | |
| EP2686310B1 | European Patent Office (EPO) | B1 | |
| DK2686310T3 | Denmark | T3 | |
| TR2018002550T4 | Türkiye | T4 | |
| TR201802550T4 | Türkiye | T4 | |
| ES2660493T3 | Spain | T3 | |
| MX355309B | Mexico | B | |
| PL2686310T3 | Poland | T3 | |
| DK2686310T5 | Denmark | T5 | |
| HUE036408T2 | Hungary | T2 | |
| KR101893756B1 | Republic of Korea | B1 | |
| CA2835617C | Canada | C | |
| BR112013023517B1 | Brazil | B1 |
Numbers
- Application
- 2013007044
Titles
- English
- Benzodioxane inhibitors of leukotriene production
Classification
- CPC, 30
- C07D405/10
- C07D295/16
- C07D405/12
- C07D405/14
- C07D487/10
- A61K31/5377
- A61K31/397
- C07D319/20
- C07D417/10
- C07D417/14
- C07D471/10
- C07D487/04
- C07D487/08
- C07D491/056
- C07D295/096
- A61P1/00
- A61P11/06
- A61P13/12
- A61P19/00
- A61P25/04
- A61P29/00
- A61P31/04
- A61P35/00
- A61P37/08
- A61P7/00
- A61P9/00
- A61P9/10
- A61P9/12
- C07D413/10
- A61K31/357
- IPC, 7
- A61K31 357
- A61P19 00
- C07D319 20
- C07D405 10
- C07D405 12
- C07D405 14
- C07D487 10