AP1905A
Pyrrolo[2,3-d] Pyrimidine Compounds.
Abstract
A compound of formula (I) wherein R1,R2 and R3 are as defined above, which are inhibitors of the enzyme protein kinases such as Janus Kinase 3 and as such are useful therapy as immunosuppressive agents for organ transplants, xeno transplantation, lupus, multiple scelerosis, rheumatoid arthritis, psoriasis, Type I diabetes and complications from diabetes, cancer, asthma, atopic dermatitis, autoimmune thyroid disorders, ulcerative colitis, Crohn's disease, Alzheimer's disease, Leukemia and other autoimmune diseases.
Term
No projected expiry on record.
- Priority
- Filed
- Granted
- Today
Every citation, both waysCites: the store holds 1 of 2
| Document | Relation | Office | Cited during |
|---|---|---|---|
| EP0795556A1 | Cites | European Patent Office (EPO) | Search report |
| J. of Med. Chem.; US Chem. Soc.; Vol.39, No.12 | Non-patent | – | Search report |
106 members in 55 offices
Priority claims7
| Document | Office | Kind | Date |
|---|---|---|---|
| 17017999 | United States of America | P | |
| 17017999 | United States of America | P | |
| 0001742 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| 0001742 | International Bureau of the World Intellectual Property Organization (WIPO) | W | |
| 60170179 | – | – | – |
| US19990170179P | – | – | – |
| WO2000IB01742 | – | – | – |
Members106
| Document | Office | Kind | |
|---|---|---|---|
| HN2000000265A | Honduras | A | |
| ECSP003819A | Ecuador | A | |
| CA2393640A1 | Canada | A1 | |
| DZ3248A1 | Algeria | A1 | |
| WO0142246A2 | World Intellectual Property Organization (WIPO) | A2 | |
| AU1295001A | Australia | A | |
| UY26477A1 | Uruguay | A1 | |
| PE20011096A1 | Peru | A1 | |
| WO0142246A3 | World Intellectual Property Organization (WIPO) | A3 | |
| US2001053782A1 | United States of America | A1 | |
| PA8507301A1 | Panama | A1 | |
| IS6383A | Iceland | A | |
| GT200000208A | Guatemala | A | |
| NO20022738D0 | Norway | D0 | |
| NO20022738L | Norway | L | |
| SV2002000236A | El Salvador | A | |
| KR20020061637A | Republic of Korea | A | |
| BR0016263A | Brazil | A | |
| MXPA02005675A | Mexico | A | |
| EP1235830A2 | European Patent Office (EPO) | A2 | |
| IL149616D0 | Israel | D0 | |
| EA200200506A1 | Eurasian Patent Organization (EAPO) | A1 | |
| BG106855A | Bulgaria | A | |
| TR200201498T2 | Türkiye | T2 | |
| AR026534A1 | Argentina | A1 | |
| HU0203503A2 | Hungary | A2 | |
| HUP0203503A2 | Hungary | A2 | |
| CN1409712A | China | A | |
| CO5271665A1 | Colombia | A1 | |
| JP2003516405A | Japan | A | |
| EE200200304A | Estonia | A | |
| CZ20021846A3 | Czechia | A3 | |
| HK1051195A1 | Hong Kong, China | A1 | |
| SK7562002A3 | Slovakia | A3 | |
| ZA200204535B | South Africa | B | |
| US6627754B2 | United States of America | B2 | |
| CR6655A | Costa Rica | A | |
| EP1235830B1 | European Patent Office (EPO) | B1 | |
| AT257157T | Austria | T | |
| ATE257157T1 | Austria | T1 | |
| EP1382339A1 | European Patent Office (EPO) | A1 | |
| DE60007552D1 | Germany | D1 | |
| TR200400105T4 | Türkiye | T4 | |
| NZ518884A | New Zealand | A | |
| US2004053947A1 | United States of America | A1 | |
| DK1235830T3 | Denmark | T3 | |
| PT1235830E | Portugal | E | |
| PL355907A1 | Poland | A1 | |
| ES2208433T3 | Spain | T3 | |
| SI1235830T1 | Slovenia | T1 | |
| HRP20020509A2 | Croatia | A2 | |
| DE60007552T2 | Germany | T2 | |
| AU777911B2 | Australia | B2 | |
| TW200427453A | Taiwan Province of China | A | |
| MA26851A1 | Morocco | A1 | |
| HU0203503A3 | Hungary | A3 | |
| HUP0203503A3 | Hungary | A3 | |
| UA72290C2 | Ukraine | C2 | |
| YU41302A | Yugoslavia, later Serbia and Montenegro (until 2006) | A | |
| KR100477818B1 | Republic of Korea | B1 | |
| NZ528905A | New Zealand | A | |
| GEP20053479B | Georgia | B | |
| CN1195755C | China | C | |
| HRP20020509B1 | Croatia | B1 | |
| US6956041B2 | United States of America | B2 | |
| EA006227B1 | Eurasian Patent Organization (EAPO) | B1 | |
| TNSN00239A1 | Tunisia | A1 | |
| US2005288313A1 | United States of America | A1 | |
| TWI248935B | Taiwan Province of China | B | |
| OA12118A | African Intellectual Property Organization (OAPI) | A | |
| US7091208B2 | United States of America | B2 | |
| CA2393640C | Canada | C | |
| TWI264305B | Taiwan Province of China | B | |
| US2006241131A1 | United States of America | A1 | |
| IS2173B | Iceland | B | |
| NO323378B1 | Norway | B1 | |
| CU23220A3 | Cuba | A3 | |
| MY130760A | Malaysia | A | |
| US7265221B2 | United States of America | B2 | |
| EP1382339B1 | European Patent Office (EPO) | B1 | |
| AT380031T | Austria | T | |
| ATE380031T1 | Austria | T1 | |
| US2007292430A1 | United States of America | A1 | |
| DE60037345D1 | Germany | D1 | |
| DK1382339T3 | Denmark | T3 | |
| PT1382339E | Portugal | E | |
| ES2295495T3 | Spain | T3 | |
| JP4078074B2 | Japan | B2 | |
| AP1905AThis record | African Regional Intellectual Property Organization (ARIPO) | A | |
| DE60037345T2 | Germany | T2 | |
| EG24399A | Egypt | A | |
| US7601727B2 | United States of America | B2 | |
| BG65821B1 | Bulgaria | B1 | |
| SK287188B6 | Slovakia | B6 | |
| US2010035903A1 | United States of America | A1 | |
| IL149616A | Israel | A | |
| USRE41783E | United States of America | E | |
| EE05351B1 | Estonia | B1 | |
| US7842699B2 | United States of America | B2 | |
| RS51574B | Serbia | B |
Showing 100 of 106
Numbers
- Publication
- AP 1905
- Publication, DOCDB
- 1905
- Publication, EPODOC
- AP1905
- Application
- 2002002543
- Application, DOCDB
- 2002002543
- Application, EPODOC
- AP20020002543
Titles
- English
- Pyrrolo[2,3-d] Pyrimidine Compounds.
Classification
- CPC, 23
- C07D487/04
- A61K31/365
- A61K31/445
- A61K31/519
- A61K31/52
- A61K31/54
- A61K31/56
- A61K38/13
- A61K45/06
- A61P1/00
- A61P1/04
- A61P11/06
- A61P17/00
- A61P17/06
- A61P19/02
- A61P25/28
- A61P29/00
- A61P35/00
- A61P35/02
- A61P37/00
- A61P37/06
- A61P43/00
- A61P3/10
- IPC, 21
- A61K31 00
- A61K31 365
- A61K31 445
- A61K31 519
- A61K38 13
- A61K45 06
- A61P1 00
- A61P1 04
- A61P3 10
- A61P11 06
- A61P17 00
- A61P17 06
- A61P25 28
- A61P29 00
- A61P35 00
- A61P35 02
- A61P37 00
- A61P37 06
- A61P43 00
- C07D487 02
- C07D487 04