Chiral salt resolution.
Abstract
A method for resolving enantiomers of a compound containing the structure of the formula: wherein r4 or r5 may contain one or more asymmetric centres, by mixing a racemic mixture of enantioners of a compound, containing the structure of said formula; in a solvent, with a resolving compound having a defined stereospecificity, to form a solution and with said resolving agent being capable of binding with at least one but not all of said enantiomers to form a precipitate, containing said at least one of said enantiomers in stereospecific form and collecting either the precipitate and purifying it or collecting the solution with contained other of said enantiomers and recrystallizing the enantiomer contained in said solution.
Term
No projected expiry on record.
- Priority
- Filed
- Granted
- Today
Every citation, both waysCites: the store holds 2 of 3
| Document | Relation | Office | Cited during |
|---|---|---|---|
| US4814477A | Cites | United States of America | Search report |
| WO9965909A1 | Cites | World Intellectual Property Organization (WIPO) | Search report |
| Jaques J: 1981, J. Willy & Sons, Inc | Non-patent | – | Search report |
| Baylea C.R. et al: 1992, J. Willy & Sons | Non-patent | – | Search report |
107 members in 53 offices
Priority claims8
| Document | Office | Kind | Date |
|---|---|---|---|
| 29477501 | United States of America | P | |
| 29477501 | United States of America | P | |
| 34104801 | United States of America | P | |
| 34104801 | United States of America | P | |
| 60294775 | – | – | – |
| 60341048 | – | – | – |
| US20010294775P | – | – | – |
| US20010341048P | – | – | – |
Members107
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|---|---|---|---|
| AP2002002550A0 | African Regional Intellectual Property Organization (ARIPO) | A0 | |
| CA2448281A1 | Canada | A1 | |
| WO02096909A1 | World Intellectual Property Organization (WIPO) | A1 | |
| GT200200100A | Guatemala | A | |
| UY27317A1 | Uruguay | A1 | |
| US2003073719A1 | United States of America | A1 | |
| PA8546301A1 | Panama | A1 | |
| PE20030561A1 | Peru | A1 | |
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| NO20035201L | Norway | L | |
| NO20093135L | Norway | L | |
| KR20040003037A | Republic of Korea | A | |
| ECSP034865A | Ecuador | A | |
| EP1392694A1 | European Patent Office (EPO) | A1 | |
| CZ20033260A3 | Czechia | A3 | |
| MXPA03011062A | Mexico | A | |
| EE200300594A | Estonia | A | |
| EA200301193A1 | Eurasian Patent Organization (EAPO) | A1 | |
| SK14652003A3 | Slovakia | A3 | |
| IL158588A0 | Israel | A0 | |
| IL158588D0 | Israel | D0 | |
| BR0209246A | Brazil | A | |
| TW200413370A | Taiwan Province of China | A | |
| ZA200307982B | South Africa | B | |
| AR037321A1 | Argentina | A1 | |
| JP2004534047A | Japan | A | |
| US2004229923A1 | United States of America | A1 | |
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| HRP20030943A2 | Croatia | A2 | |
| AR045680A2 | Argentina | A2 | |
| TNSN03128A1 | Tunisia | A1 | |
| EP1609781A1 | European Patent Office (EPO) | A1 | |
| CN1729192A | China | A | |
| KR20060014459A | Republic of Korea | A | |
| GEP20063784B | Georgia | B | |
| EP1666481A2 | European Patent Office (EPO) | A2 | |
| OA12612A | African Intellectual Property Organization (OAPI) | A | |
| YU92303A | Yugoslavia, later Serbia and Montenegro (until 2006) | A | |
| EA007251B1 | Eurasian Patent Organization (EAPO) | B1 | |
| EA200600575A1 | Eurasian Patent Organization (EAPO) | A1 | |
| EP1666481A3 | European Patent Office (EPO) | A3 | |
| KR20060133117A | Republic of Korea | A | |
| MY129649A | Malaysia | A | |
| NZ540332A | New Zealand | A | |
| GT200200100AA | Guatemala | A | |
| HU0400152A2 | Hungary | A2 | |
| HUP0400152A2 | Hungary | A2 | |
| UA80093C2 | Ukraine | C2 | |
| US7301023B2 | United States of America | B2 | |
| KR20080002931A | Republic of Korea | A | |
| AU2002304401B2 | Australia | B2 | |
| AP1859AThis record | African Regional Intellectual Property Organization (ARIPO) | A | |
| CL2008000762A1 | Chile | A1 | |
| AU2008203170A1 | Australia | A1 | |
| CR10177A | Costa Rica | A | |
| KR20080083028A | Republic of Korea | A | |
| US7432370B2 | United States of America | B2 | |
| KR100868814B1 | Republic of Korea | B1 | |
| KR100869409B1 | Republic of Korea | B1 | |
| CU23337B7 | Cuba | B7 | |
| AU2002304401C1 | Australia | C1 | |
| CA2448281C | Canada | C | |
| TWI310384B | Taiwan Province of China | B | |
| AU2008203170B2 | Australia | B2 | |
| TWI316061B | Taiwan Province of China | B | |
| KR100926875B1 | Republic of Korea | B1 | |
| JP4381137B2 | Japan | B2 | |
| EA012666B1 | Eurasian Patent Organization (EAPO) | B1 | |
| NO328578B1 | Norway | B1 | |
| EE05332B1 | Estonia | B1 | |
| EP1609781B1 | European Patent Office (EPO) | B1 | |
| AT519741T | Austria | T | |
| ATE519741T1 | Austria | T1 | |
| ES2369226T3 | Spain | T3 | |
| HRP20030943B1 | Croatia | B1 | |
| RS52144B | Serbia | B | |
| EP1666481B1 | European Patent Office (EPO) | B1 | |
| DK1666481T3 | Denmark | T3 | |
| SI1666481T1 | Slovenia | T1 | |
| PT1666481E | Portugal | E | |
| ES2393385T3 | Spain | T3 | |
| HU0400152A3 | Hungary | A3 | |
| HUP0400152A3 | Hungary | A3 | |
| EP1666481B9 | European Patent Office (EPO) | B9 | |
| CZ304366B6 | Czechia | B6 | |
| SK288192B6 | Slovakia | B6 | |
| SK288199B6 | Slovakia | B6 | |
| PL409305A1 | Poland | A1 | |
| BG66489B1 | Bulgaria | B1 | |
| CY1113322T1 | Cyprus | T1 | |
| LUC00031I1 | Luxembourg | I1 | |
| NL300887I2 | Netherlands (Kingdom of the) | I2 | |
| NO2017047I1 | Norway | I1 | |
| LTPA2017025I1 | Lithuania | I1 | |
| LUC00031I2 | Luxembourg | I2 | |
| FR17C1031I1 | France | I1 |
Numbers
- Publication
- AP 1859
- Publication, DOCDB
- 1859
- Publication, EPODOC
- AP1859
- Application
- 2550
- Application, DOCDB
- 2002002550
- Application, EPODOC
- AP20020002550
Titles
- English
- Chiral salt resolution.
Classification
- CPC, 19
- C07D487/04
- C07B2200/07
- C07D211/56
- A61P1/04
- A61P11/06
- A61P17/00
- A61P17/06
- A61P19/02
- A61P25/00
- A61P25/28
- A61P29/00
- A61P35/00
- A61P35/02
- A61P37/00
- A61P37/02
- A61P37/06
- A61P37/08
- A61P43/00
- A61P3/10
- IPC, 24
- A61K31 505
- A61K
- A61K31 519
- A61K45 00
- A61P
- A61P1 04
- A61P3 10
- A61P11 06
- A61P17 00
- A61P17 06
- A61P19 02
- A61P25 00
- A61P25 28
- A61P29 00
- A61P35 00
- A61P35 02
- A61P37 02
- A61P37 06
- A61P37 08
- A61P43 00
- C07B57 00
- C07D
- C07D211 56
- C07D487 04